Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Liver carboxylesterase (Sus scrofa) | BDBM50570559 (CHEMBL4868687) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Competitive inhibition of porcine liver carboxylesterase by double reciprocal Lineweaver-Burk plot analysis | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50300582 (CHEMBL573979 | Dibutyl 2,2,2-trifluoro-1-phenyleth...) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 156 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase by Lineweaver-Burk analysis | Bioorg Med Chem Lett 19: 5528-30 (2009) Article DOI: 10.1016/j.bmcl.2009.08.065 BindingDB Entry DOI: 10.7270/Q2VH5NXD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50267978 (CHEMBL4096931) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 230 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Postovsky Institute of Organic Synthesis, Urals Branch of Russian Academy of Sciences, Yekaterinburg 620990, Russia. Curated by ChEMBL | Assay Description Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed... | Bioorg Med Chem 25: 3997-4007 (2017) Article DOI: 10.1016/j.bmc.2017.05.045 BindingDB Entry DOI: 10.7270/Q2F76G21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50529195 (CHEMBL4475685) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 337 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ural Branch of Russian Academy of Sciences Curated by ChEMBL | Assay Description Competitive inhibition of porcine liver carboxylesterase by double reciprocal Lineweaver-Burk plot analysis | Bioorg Med Chem Lett 29: (2019) Article DOI: 10.1016/j.bmcl.2019.126716 BindingDB Entry DOI: 10.7270/Q2CR5XTF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50500766 (CHEMBL3754409) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre... | Bioorg Med Chem 24: 1050-62 (2016) Article DOI: 10.1016/j.bmc.2016.01.031 BindingDB Entry DOI: 10.7270/Q2B85C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50500752 (CHEMBL3754327) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 440 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre... | Bioorg Med Chem 24: 1050-62 (2016) Article DOI: 10.1016/j.bmc.2016.01.031 BindingDB Entry DOI: 10.7270/Q2B85C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50268001 (CHEMBL4100446) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 570 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Postovsky Institute of Organic Synthesis, Urals Branch of Russian Academy of Sciences, Yekaterinburg 620990, Russia. Curated by ChEMBL | Assay Description Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed... | Bioorg Med Chem 25: 3997-4007 (2017) Article DOI: 10.1016/j.bmc.2017.05.045 BindingDB Entry DOI: 10.7270/Q2F76G21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50267979 (CHEMBL4069738) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Postovsky Institute of Organic Synthesis, Urals Branch of Russian Academy of Sciences, Yekaterinburg 620990, Russia. Curated by ChEMBL | Assay Description Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed... | Bioorg Med Chem 25: 3997-4007 (2017) Article DOI: 10.1016/j.bmc.2017.05.045 BindingDB Entry DOI: 10.7270/Q2F76G21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50267977 (CHEMBL4080436) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Postovsky Institute of Organic Synthesis, Urals Branch of Russian Academy of Sciences, Yekaterinburg 620990, Russia. Curated by ChEMBL | Assay Description Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed... | Bioorg Med Chem 25: 3997-4007 (2017) Article DOI: 10.1016/j.bmc.2017.05.045 BindingDB Entry DOI: 10.7270/Q2F76G21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50500755 (CHEMBL3752466) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre... | Bioorg Med Chem 24: 1050-62 (2016) Article DOI: 10.1016/j.bmc.2016.01.031 BindingDB Entry DOI: 10.7270/Q2B85C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50300581 (CHEMBL575301 | Diethyl 2,2,2-trifluoro-1-phenyleth...) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase by Lineweaver-Burk analysis | Bioorg Med Chem Lett 19: 5528-30 (2009) Article DOI: 10.1016/j.bmcl.2009.08.065 BindingDB Entry DOI: 10.7270/Q2VH5NXD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50500757 (CHEMBL3752682) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre... | Bioorg Med Chem 24: 1050-62 (2016) Article DOI: 10.1016/j.bmc.2016.01.031 BindingDB Entry DOI: 10.7270/Q2B85C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50267981 (CHEMBL4089864) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 6.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Postovsky Institute of Organic Synthesis, Urals Branch of Russian Academy of Sciences, Yekaterinburg 620990, Russia. Curated by ChEMBL | Assay Description Competitive inhibition of porcine liver carboxylesterase using varying levels of 4-nitrophenol acetate as substrate preincubated for 10 mins followed... | Bioorg Med Chem 25: 3997-4007 (2017) Article DOI: 10.1016/j.bmc.2017.05.045 BindingDB Entry DOI: 10.7270/Q2F76G21 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50300580 (CHEMBL575281 | Dimethyl 2,2,2-trifluoro-1-phenylet...) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.64E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase by Lineweaver-Burk analysis | Bioorg Med Chem Lett 19: 5528-30 (2009) Article DOI: 10.1016/j.bmcl.2009.08.065 BindingDB Entry DOI: 10.7270/Q2VH5NXD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50500758 (CHEMBL3753216) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 7.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre... | Bioorg Med Chem 24: 1050-62 (2016) Article DOI: 10.1016/j.bmc.2016.01.031 BindingDB Entry DOI: 10.7270/Q2B85C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50500748 (CHEMBL3753156) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | 7.81E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institute of Physiologically Active Compounds Russian Academy of Sciences Curated by ChEMBL | Assay Description Noncompetitive inhibition of porcine liver carboxylesterase using 4-nitrophenol acetate as substrate assessed as steady state inhibition constant pre... | Bioorg Med Chem 24: 1050-62 (2016) Article DOI: 10.1016/j.bmc.2016.01.031 BindingDB Entry DOI: 10.7270/Q2B85C4Q | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50409669 (CHEMBL155514) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.457 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description In vitro inhibition of porcine carboxylesterase. | J Med Chem 45: 5576-93 (2002) BindingDB Entry DOI: 10.7270/Q2DN4671 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371969 (CHEMBL270374) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371971 (CHEMBL440542) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371969 (CHEMBL270374) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371970 (CHEMBL89506) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL DrugBank PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371966 (CHEMBL269931) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371973 (CHEMBL402615) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570553 (CHEMBL4854298) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570555 (CHEMBL4868014) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371972 (CHEMBL270375) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371966 (CHEMBL269931) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371970 (CHEMBL89506) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL DrugBank PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570549 (CHEMBL4853742) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570554 (CHEMBL4858186) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.20 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570551 (CHEMBL4853637) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570550 (CHEMBL4849361) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371971 (CHEMBL440542) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570561 (CHEMBL4855838) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371971 (CHEMBL440542) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.32 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description In vitro inhibition of porcine carboxylesterase. | J Med Chem 45: 5576-93 (2002) BindingDB Entry DOI: 10.7270/Q2DN4671 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371968 (CHEMBL273138) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.60 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371959 (CHEMBL86668) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.30 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50409660 (CHEMBL155513) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 10.5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description In vitro inhibition of porcine carboxylesterase. | J Med Chem 45: 5576-93 (2002) BindingDB Entry DOI: 10.7270/Q2DN4671 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371972 (CHEMBL270375) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371968 (CHEMBL273138) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570552 (CHEMBL4855755) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50409672 (CHEMBL153080) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 17.0 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description In vitro inhibition of porcine carboxylesterase. | J Med Chem 45: 5576-93 (2002) BindingDB Entry DOI: 10.7270/Q2DN4671 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371973 (CHEMBL402615) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371961 (CHEMBL270373) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371959 (CHEMBL86668) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50570559 (CHEMBL4868687) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of porcine liver carboxylesterase using 4-NPA as substrate preincubated for 10 mins followed by substrate addition by spectrophotometric a... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113385 BindingDB Entry DOI: 10.7270/Q2FJ2MK0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371965 (CHEMBL272075) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371962 (CHEMBL155396) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 33 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 15 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371967 (CHEMBL257071) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description Inhibition of pig liver carboxylesterase after 5 mins | Bioorg Med Chem 16: 2114-30 (2008) Article DOI: 10.1016/j.bmc.2007.10.081 BindingDB Entry DOI: 10.7270/Q2K938DT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Liver carboxylesterase (Sus scrofa) | BDBM50371970 (CHEMBL89506) | PDB KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL DrugBank PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
University of California at Davis Curated by ChEMBL | Assay Description Inhibition of Sus scrofa (pig) carboxylesterase isolated from liver in using p-nitrophenyl acetate as substrate incubated for 5 min prior to substrat... | Chem Res Toxicol 14: 1563-72 (2001) Article DOI: 10.1021/tx015508+ BindingDB Entry DOI: 10.7270/Q20004ZT | |||||||||||
More data for this Ligand-Target Pair |
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