Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily KQT member 4 (Rattus norvegicus) | BDBM50121051 (CHEMBL3621437) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 376 | n/a | n/a | n/a | n/a |
Pfizer Inc. Curated by ChEMBL | Assay Description Activation of rat Kv7.4 expressed in CHOK1 cells | Bioorg Med Chem Lett 25: 4941-4 (2015) Article DOI: 10.1016/j.bmcl.2015.04.074 BindingDB Entry DOI: 10.7270/Q28054FG | |||||||||||
More data for this Ligand-Target Pair |