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BindingDB Data by Journal

PMIDDataArticle TitleCitationOrganizationSD Files Download
27894870141A benzo[b]thiophene-based selective type 4 S1P receptor agonist.EBIBioorg Med Chem Lett 27: 1-5 (2017)Harvard Medical School2D 3D TSV
2789037820Design and synthesis of 4,5,6,7-tetrahydro-1H-1,2-diazepin-7-one derivatives as a new series of Phosphodiesterase 4 (PDE4) inhibitors.EBIBioorg Med Chem Lett 27: 24-29 (2017)University of Genoa2D 3D TSV
278903812Evaluation of dipeptide nitriles as inhibitors of rhodesain, a major cysteine protease of Trypanosoma brucei.EBIBioorg Med Chem Lett 27: 45-50 (2017)Johannes Gutenberg-University2D 3D TSV
2787647568Microwave assisted synthesis of novel tetrazole/sulfonamide derivatives based on octahydroacridine, xanthene and chromene skeletons as inhibitors of the carbonic anhydrases isoforms I, II, IV and VII.EBIBioorg Med Chem Lett 27: 86-89 (2017)Dumlupinar University2D 3D TSV
2789487411MARK inhibitors: Declaring a No-Go decision on a chemical series based on extensive DMPK experimentation.EBIBioorg Med Chem Lett 27: 109-113 (2017)Merck& Co.2D 3D TSV
27816515143Structure guided design of a series of selective pyrrolopyrimidinone MARK inhibitors.EBIBioorg Med Chem Lett 27: 114-120 (2017)Merck& Co.2D 3D TSV
2797959573Imidazopyridyl compounds as aldosterone synthase inhibitors.EBIBioorg Med Chem Lett 27: 143-146 (2017)Merck USA2D 3D TSV
2793917484Challenges in the development of an MEBIBioorg Med Chem Lett 27: 171-175 (2017)Vanderbilt University Medical Center2D 3D TSV
2796488123Bivalent SIRT1 inhibitors.EBIBioorg Med Chem Lett 27: 180-186 (2017)Jiangsu University2D 3D TSV
2792361770Novel pyrazolo[1,5-a]pyridines with improved aqueous solubility as p110a-selective PI3 kinase inhibitors.EBIBioorg Med Chem Lett 27: 187-190 (2017)University of Auckland2D 3D TSV
2792361835Novel 3-methylindoline inhibitors of EZH2: Design, synthesis and SAR.EBIBioorg Med Chem Lett 27: 217-222 (2017)Integral BioSciences Pvt. Ltd.2D 3D TSV
2791479614Design and synthesis of new piperidone grafted acetylcholinesterase inhibitors.EBIBioorg Med Chem Lett 27: 228-231 (2017)University of Nebraska Medical Center2D 3D TSV
2792361913Synthesis and application of฿-carbolines as novel multi-functional anti-Alzheimer's disease agents.EBIBioorg Med Chem Lett 27: 232-236 (2017)University of Massachusetts Boston2D 3D TSV
2791480212Synthesis and in vitro antiproliferative activity of C5-benzyl substituted 2-amino-pyrrolo[2,3-d]pyrimidines as potent Hsp90 inhibitors.EBIBioorg Med Chem Lett 27: 237-241 (2017)Korea University2D 3D TSV
279131825Virtual screening and biophysical studies lead to HSP90 inhibitors.EBIBioorg Med Chem Lett 27: 277-281 (2017)University of Auckland2D 3D TSV
2791480011Discovery of a new isomannide-based peptidomimetic synthetized by Ugi multicomponent reaction as human tissue kallikrein 1 inhibitor.EBIBioorg Med Chem Lett 27: 314-318 (2017)Universidade Federal Fluminense2D 3D TSV
2790876155Discovery of dual positive allosteric modulators (PAMs) of the metabotropic glutamate 2 receptor and CysLT1 antagonists for treating migraine headache.EBIBioorg Med Chem Lett 27: 323-328 (2017)Eli Lilly and Company2D 3D TSV
278992653Discovery of novel DNA methyltransferase 3A inhibitors via structure-based virtual screening and biological assays.EBIBioorg Med Chem Lett 27: 342-346 (2017)University of Science and Technology of China2D 3D TSV
2791965724Synthesis of novel steroidal agonists, partial agonists, and antagonists for the glucocorticoid receptor.EBIBioorg Med Chem Lett 27: 347-353 (2017)The Scripps Research Institute2D 3D TSV