Compound Name
(alphabetical) | Enz. Inhib. Data | ITC Data | Binding Targets | Alternate Compound Names |
|---|
| Ki | IC50 | Kd | EC50 | Koff | Kon | Other |
|---|
BDBM48320
 | 59 | 23 | 2 | 4 | 0 | 0 | 0 | 0 | - 5-HT3A Serotonin Receptor
- 5-hydroxytryptamine receptor 1A (5-HT1A)
- 5-hydroxytryptamine receptor 4 (5-HT4)
- 6-phosphogluconate dehydrogenase (6PGD)
- ADRB2
- Acetylcholinesterase
- Adrenergic Alpha
- Adrenergic receptor alpha-2
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Bile salt export pump
- Cytochrome P450 2D6 (2D6)
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- DOPAMINE
- DRD2
- Dopamine D2 receptor and Serotonin 2a receptor (D2 and 5HT2a)
- Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor
- Dopamine receptor
- Estradiol receptor beta (ERβ)
- HTR4
- HTR6
- Histamine H1 receptor
- Lactoperoxidase (LPO)
- Muscarinic acetylcholine receptor M2
- Myeloperoxidase
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin 3 receptor (5HT3)
- Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
- Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
- Serum albumin
- adrenergic Alpha2
| - 4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-methoxy-benzamide;hydrochloride
- 4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-methoxybenzamide;hydrochloride
- 4-azanyl-5-chloranyl-N-[2-(diethylamino)ethyl]-2-methoxy-benzamide;hydrochloride
- METOCLOPRAMIDE
- METOCLOPRAMIDE HYDROCHLORIDE
- MLS000069667
- Metochloropramide
- SMR000058471
- US9132134, Metoclopramide
- cid_23659
|
BDBM50005836
 | 48 | 38 | 0 | 2 | 0 | 0 | 0 | 0 | - 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 4 (5-HT4)
- Adrenergic receptor alpha
- Adrenergic receptor alpha-1
- Adrenergic receptor alpha-2
- Adrenergic receptor beta
- Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor
- Alpha-1A adrenergic receptor
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor and beta-3 adrenergic receptor
- D(1A) dopamine receptor
- D(2) dopamine receptor
- DOPAMINE
- Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor
- HTR4
- HTR6
- Potassium voltage-gated channel subfamily H member 2
- Serotonin (5-HT) receptor
- Serotonin 1 (5-HT1) receptor
- Serotonin 2 (5-HT2) receptor
- Serotonin 2a (5-HT2a) receptor
- Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
- Serotonin 3a (5-HT3a)/3b (5-HT3b)/3c (5-HT3c)/3d (5-HT3d)/3e (5-HT3e) receptor
- Serotonin receptor (2b and 2c)
- Serotonin receptor 2a and 2b (5HT2A and 5HT2B)
- Sodium channel protein type 5 subunit alpha
- Voltage-dependent L-type calcium channel subunit alpha-1C
- ubiquitin-conjugating enzyme E2 N
| - 4-Amino-5-chloro-N-{1-[3-(4-fluoro-phenoxy)-propyl]-3-methoxy-piperidin-4-yl}-2-methoxy-benzamide
- 4-amino-5-chloro-N-(1-(3-(4-fluorophenoxy)propyl)-3-methoxypiperidin-4-yl)-2-methoxybenzamide
- CHEMBL560739
- CISAPRIDE
- PROPULSID
- US10167299, Cisapride
- US9221790, Cisapride
- cid_5311047
|
BDBM50171290
 | 88 | 0 | 0 | 0 | 0 | 0 | 0 | 0 | - 5-Hydroxytryptamine receptor 7 (5-HT7)
- 5-hydroxytryptamine receptor 1B
- 5-hydroxytryptamine receptor 1D
- 5-hydroxytryptamine receptor 2A
- 5-hydroxytryptamine receptor 2C
- 5-hydroxytryptamine receptor 3A
- 5-hydroxytryptamine receptor 4 (5-HT4)
- ADORA3
- ATP-sensitive inward rectifier potassium channel 1
- AVPR1A
- Adenosine receptor A1
- Adenosine receptor A2
- Alpha-1A adrenergic receptor
- Alpha-2A adrenergic receptor
- Alpha-2B adrenergic receptor
- Alpha-2C adrenergic receptor
- Angiotensin II AT2
- Angiotensin II receptor
- Benzodiazepine central
- Benzodiazepine peripheral
- Beta-1 adrenergic receptor
- Beta-2 adrenergic receptor and beta-3 adrenergic receptor
- CHRM5
- Calcitonin gene-related peptide (CGRP alpha)
- Calcium channel (DHP)
- Calcium channel (Type L)
- Cannabinoid receptor 1
- Cannabinoid receptor 2
- Chloride channel, TBOB
- Cholecystokinin receptor
- Cysteinyl leukotriene receptor 1
- D(1A) dopamine receptor
- D(2) dopamine receptor
- D(3) dopamine receptor
- Disintegrin and metalloproteinase domain-containing protein 17
- Dopamine D5 receptor
- Dopamine receptors; D2 & D4
- EDNRB
- Endothelin-1 receptor
- GALANIN
- GRIA3
- GRIK1
- GRPR
- Gamma-aminobutyric acid type B receptor subunit 1
- Glucocorticoid receptor
- Glutamate receptor ionotropic, NMDA 1
- Glycine, non-strychnine
- HTR6
- Histamine H1 receptor
- Histamine H2 Receptor
- Histamine receptor (H3)
- Imidazoline receptor 1 (I1R)
- Kappa-type opioid receptor
- Leukotriene 2
- Melatonin receptor
- Muscarinic acetylcholine receptor M1
- Muscarinic acetylcholine receptor M2
- Muscarinic acetylcholine receptor M3
- Muscarinic acetylcholine receptor M4
- NMBR
- NT
- Neuromedin-K receptor
- Neuropeptide Y receptor type 1
- Neuropeptide Y receptor type 2
- Nociceptin/mu opioid receptor
- P2X purinoceptor 1
- Platelet activating factor receptor
- Potassium Channel (Ca2+ dependent)
- Prostaglandin G/H synthase (cyclooxygenase)
- Purinergic receptor P2Y1
- SOMATOSTATIN
- Serotonin (5-HT) receptor
- Sigma-1
- Substance-K receptor
- Substance-P receptor
- VIP peptides
- Vasopressin V2 receptor (V2)
- Voltage-gated calcium channel subunit alpha Cav2.2
- Voltage-gated potassium channel
- Voltage-gated sodium channel subunit alpha Nav1.1 (Nav1.1)
- Voltage-gated sodium channel subunit alpha Nav1.2 (Nav1.2)
| - 5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide
- CHEMBL189676
- SR 147778
|
BDBM50380399
 | 3 | 85 | 0 | 0 | 0 | 0 | 0 | 0 | - Histone Deacetylase 10 (HDAC10)
- Histone deacetylase 1
- Histone deacetylase 1/2/3
- Histone deacetylase 11
- Histone deacetylase 2
- Histone deacetylase 3
- Histone deacetylase 3/Nuclear receptor corepressor 2
- Histone deacetylase 4
- Histone deacetylase 5
- Histone deacetylase 6
- Histone deacetylase 7
- Histone deacetylase 8
- Histone deacetylase 9
| - CHEMBL2018302
- Tubastatin A
- US8748451, 6
- US9249087, Tubacin
- US9751832, Tubastatin A
|
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