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Targets Binding with 1093 Compounds


Target NameCommercially
Available
Compounds
Protein/Small MoleculeOther

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AffyNet
KiIC50KdEC50koffkonotherITCSDFTSV
1 ACAT-related gene product 1BDB 0 17 1216 0 43 0 0 0 0 0 40 5 2D 3DTSV
2 Cytosolic NADP-isocitrate dehydrogenaseBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
3 Diacylglycerol Acyltransferase (DGAT1)BDB 0 17 1216 0 43 0 0 0 0 0 40 5 2D 3DTSV
4 Diacylglycerol O-acyltransferase 1BDB 11 17 1486 0 43 0 0 0 0 0 41 8 2D 3DTSV
5 Diacylglycerol O-acyltransferase 1 (DGAT1)BDB 8 17 1457 0 43 0 0 0 0 0 40 7 2D 3DTSV
6 Diglyceride acyltransferaseBDB 11 17 1486 0 43 0 0 0 0 0 41 8 2D 3DTSV
7 IDHBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
8 IDH1BDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
9 IDPBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
10 Isocitrate Dehydrogenase (IDH1)BDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
11 Isocitrate dehydrogenase (IDH1)(WT)BDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
12 Isocitrate dehydrogenase 1 (IDH1)BDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
13 Isocitrate dehydrogenase 1 (IDH1)(R132H)BDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
14 Isocitrate dehydrogenase [NADP] cytoplasmicBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
15 NADP(+)-specific ICDHBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
16 Oxalosuccinate decarboxylaseBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
17 PICDBDB 9 138 1682 3 0 0 0 0 0 0 10 8 2D 3DTSV
Sub total1381741270453621500000
Total29037