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Targets Binding with 1144 Compounds


Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Pyruvate dehydrogenase kinase 1 (PDK1)
Ki: 29 IC50: 188 Kd: 25
47
7
2D 3D TSV 
Pyruvate dehydrogenase kinase isoenzyme 1 (PDK1)
Ki: 42 IC50: 1192 Kd: 179 EC50: 26 ITC: 2
115
13
2D 3D TSV 
Pyruvate dehydrogenase kinase isoform 1
Ki: 29 IC50: 188 Kd: 25
47
7
2D 3D TSV