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Targets Binding with 191 Compounds


Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Epidermal growth factor receptor (EGFR)(T790)
IC50: 93
6
0
2D 3D TSV 
Epidermal growth factor receptor (EGFR)(T790M)
IC50: 93
6
0
2D 3D TSV 
Epidermal growth factor receptor (T790M)
IC50: 93
6
0
2D 3D TSV 
Neuronal acetylcholine receptor protein beta-4 subunit
Ki: 8
1
3
2D 3D TSV 
Neuronal acetylcholine receptor subunit beta-4
Ki: 8
1
3
2D 3D TSV 
Phosphodiesterase 10A (PDE10A)
IC50: 197
3
0
2D 3D TSV 
Pyruvate dehydrogenase kinase
Ki: 30 IC50: 204 Kd: 25
49
8
2D 3D TSV 
Pyruvate dehydrogenase kinase 4 (PDK4)
Ki: 1 IC50: 16
7
1
2D 3D TSV 
Pyruvate dehydrogenase kinase isoform 4
Ki: 1 IC50: 16
7
1
2D 3D TSV 
SMO
IC50: 263 EC50: 25
13
1
2D 3D TSV