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Targets Binding with 2920 Compounds


Target NameCommercially
Available
Compounds
Protein/Small MoleculeOther

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AffyNet
KiIC50KdEC50koffkonotherITCSDFTSV
1 ARK1BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
2 AURKABDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
3 Aurora kinase A (AURA)BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
4 Aurora kinase A (AURKA)BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
5 Aurora kinase A (Aurora A)BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
6 Aurora kinase A (Aurora-2)BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
7 Aurora kinase A/Targeting protein for Xklp2BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
8 aurora-2BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
9 Aurora-related kinase 1BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
10 Breast tumor-amplified kinaseBDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
11 Breast-tumor-amplified kinaseBDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
12 BTAKBDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
13 hARK1BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
14 Serine/threonine kinase 15BDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
15 Serine/threonine-protein kinase AuroraBDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
16 Serine/threonine-protein kinase aurora ABDB 204 203 2949 235 3 0 0 1 10 0 250 7 2D 3DTSV
Sub total326432484718437604800161600
Total54256