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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
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Source Organism
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/
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Targets Binding with 301 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
β-Ketoacyl-acyl carrier protein (ACP) synthase III (FabH)
IC50:
178
6
6
2D
3D
TSV
3-oxoacyl-[acyl-carrier-protein] synthase
Ki:
36
IC50:
311
Kd:
9
15
7
2D
3D
TSV
3-oxoacyl-[acyl-carrier-protein] synthase III
Ki:
36
IC50:
412
Kd:
9
17
13
2D
3D
TSV
BDTK
IC50:
1
1
7
2D
3D
TSV
beta-Ketoacyl-ACP Synthase III (FabH)
IC50:
101
2
7
2D
3D
TSV
Brain-derived tau kinase
IC50:
1
1
7
2D
3D
TSV
Cancer/testis antigen 72
IC50:
1
1
5
2D
3D
TSV
CDK6
Ki:
1
IC50:
303
20
3
2D
3D
TSV
CDKN6
Ki:
1
IC50:
303
20
3
2D
3D
TSV
Cell division protein kinase 6
Ki:
1
IC50:
303
20
3
2D
3D
TSV
CT72
IC50:
1
1
5
2D
3D
TSV
Cyclin-dependent kinase 6
Ki:
1
IC50:
303
20
3
2D
3D
TSV
Cyclin-dependent kinase 6 (CDK 6)
Ki:
1
IC50:
303
20
3
2D
3D
TSV
Ileal bile acid transporter
Ki:
46
IC50:
291
12
4
2D
3D
TSV
KIAA0847
IC50:
1
1
5
2D
3D
TSV
KIAA1855
IC50:
1
1
7
2D
3D
TSV
Serine/threonine-protein kinase PLSTIRE
Ki:
1
IC50:
303
20
3
2D
3D
TSV
Serine/threonine-protein kinase SSTK
IC50:
1
1
5
2D
3D
TSV
Small serine/threonine kinase
IC50:
1
1
5
2D
3D
TSV
Sodium-dependent bile acid transporter (iBAT)
Ki:
46
IC50:
291
12
4
2D
3D
TSV
SSTK
IC50:
1
1
5
2D
3D
TSV
Tau-tubulin kinase 1
IC50:
1
1
7
2D
3D
TSV
Tau-tubulin kinase 2
IC50:
1
1
5
2D
3D
TSV
Testis-specific kinase 6
IC50:
1
1
5
2D
3D
TSV
Testis-specific serine/threonine-protein kinase 6
IC50:
1
1
5
2D
3D
TSV
TSK-6
IC50:
1
1
5
2D
3D
TSV
TSSK-6
IC50:
1
1
5
2D
3D
TSV
TSSK6
IC50:
1
1
5
2D
3D
TSV
TTBK1
IC50:
1
1
7
2D
3D
TSV
TTBK2
IC50:
1
1
5
2D
3D
TSV