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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
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FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
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/
Targets
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PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
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All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
Enter Data
Deposition
Contribute data
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Targets Binding with 3084 Compounds
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AffyNet
Ki
IC50
Kd
EC50
k
off
k
on
other
ITC
SDF
TSV
1
(ARTD1 or PARP1)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
2
(ARTD4 or PARP4)
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
3
(ARTD7 or PARP15)
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
4
(ARTD7 or PARP15, Y598L)
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
5
(ARTD8 or PARP14)
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
6
(ARTD8 or PARP14, Y1660L)
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
7
193 kDa vault protein
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
8
ADP-ribosyltransferase diphtheria toxin-like 1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
9
ADP-ribosyltransferase diphtheria toxin-like 12
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
10
ADP-ribosyltransferase diphtheria toxin-like 4
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
11
ADP-ribosyltransferase diphtheria toxin-like 7
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
12
ADP-ribosyltransferase diphtheria toxin-like 8
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
13
ADPRT
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
14
ADPRT 1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
15
ADPRTL1
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
16
ARTD1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
17
ARTD12
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
18
ARTD4
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
19
ARTD7
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
20
ARTD8
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
21
B aggressive lymphoma protein 2
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
22
B-aggressive lymphoma protein 3
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
23
BAL2
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
24
BAL2
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
25
BAL3
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
26
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD1 or PARP1)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
27
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD4 or PARP4)
1
0
10
0
0
0
0
0
0
0
5
6
2D
3D
TSV
28
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD7 or PARP15)
4
0
33
0
0
0
0
0
0
0
4
4
2D
3D
TSV
29
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD7 or PARP15, Y598L)
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
30
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD8 or PARP14)
3
0
20
2
0
0
0
0
0
0
4
8
2D
3D
TSV
31
Human diphtheria toxin-like ADP-ribosyltransferase (ARTD8 or PARP14, Y1660L)
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
32
KIAA0177
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
33
KIAA1268
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
34
NAD(+) ADP-ribosyltransferase 1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
35
PARP-1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
36
PARP-12
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
37
PARP-14
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
38
PARP-15
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
39
PARP-4
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
40
PARP-related/IalphaI-related H5/proline-rich
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
41
PARP1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
42
PARP12
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
43
PARP14
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
44
PARP15
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
45
PARP4
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
46
PARPL
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
47
PH5P
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
48
Poly [ADP-ribose] polymerase (PARP)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
49
Poly [ADP-ribose] polymerase 1 (PARP)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
50
Poly [ADP-ribose] polymerase 1 (PARP-1)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
51
Poly [ADP-ribose] polymerase 12
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
52
Poly [ADP-ribose] polymerase 14
3
0
19
2
0
0
0
0
0
0
3
8
2D
3D
TSV
53
Poly [ADP-ribose] polymerase 15
4
0
32
0
0
0
0
0
0
0
3
4
2D
3D
TSV
54
Poly [ADP-ribose] polymerase 4
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
55
Poly(ADP-ribose) polymerase 1 (PARP1)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
56
Poly(ADP-ribose) polymerase-1 (ARTD1/PARP1)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
57
poly-ADP-ribose polymerase 1 (PARP1)
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
58
Poly[ADP-ribose] synthase 1
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
59
PPOL
171
1168
2216
147
279
0
0
0
0
0
116
4
2D
3D
TSV
60
Vault poly(ADP-ribose) polymerase
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
61
VPARP
1
0
9
0
0
0
0
0
0
0
4
6
2D
3D
TSV
62
ZC3HDC1
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
63
Zinc finger CCCH domain-containing protein 1
0
0
2
0
0
0
0
0
0
0
1
5
2D
3D
TSV
Sub total
3005
19856
38423
2525
4743
0
0
0
0
0
Total
65547