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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
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Author
Journal/Citation
Institution
PubMed
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PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
PubMed
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All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
Enter Data
Deposition
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Targets Binding with 3467 Compounds
Target Name
Commercially
Available
Compounds
Protein/Small Molecule
Other
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UniProtKB/
Swiss-Prot/TrEMBL
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AffyNet
Ki
IC50
Kd
EC50
k
off
k
on
other
ITC
SDF
TSV
1
AIM-1
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
2
Aurora B kinase (aurB)
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
3
Aurora B-INCENP
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
4
Aurora B/Incenp
0
0
14
0
0
0
0
0
0
0
2
2
2D
3D
TSV
5
Aurora kinase 2
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
6
Aurora kinase A/B
246
380
4640
438
60
0
0
2
13
0
317
19
2D
3D
TSV
7
Aurora kinase B (AURKB)
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
8
Aurora kinase B/Inner centromere protein
158
177
1705
203
57
0
0
1
3
0
188
14
2D
3D
TSV
9
Aurora-related kinase 2
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
10
Serine/threonine-protein kinase aurora B
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
11
Serine/threonine-protein kinase Aurora-B
158
177
1691
203
57
0
0
1
3
0
186
13
2D
3D
TSV
12
STK-1
158
177
1691
249
57
0
0
1
3
0
186
13
2D
3D
TSV
Sub total
1826
2150
21578
2514
630
0
0
12
43
0
Total
26884