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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
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85%
100%
Seq ID
UniProtKB/Swiss-Prot
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Deposition
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Targets Binding with 388 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
2''''-O-methyltransferase
Ki:
36
IC50:
150
12
9
2D
3D
TSV
3.1.13.-
Ki:
36
IC50:
150
12
9
2D
3D
TSV
3C-like proteinase (3CL-PRO)
Ki:
36
IC50:
150
12
9
2D
3D
TSV
3C-like proteinase (SARS-CoV 3Cpro)
Ki:
36
IC50:
150
12
9
2D
3D
TSV
ExoN
Ki:
36
IC50:
150
12
9
2D
3D
TSV
glutamate receptor, metabotropic 3 precursor
Ki:
18
IC50:
390
EC50:
88
21
1
2D
3D
TSV
Guanine-N7 methyltransferase
Ki:
36
IC50:
150
12
9
2D
3D
TSV
Hel
Ki:
36
IC50:
150
12
9
2D
3D
TSV
Helicase
Ki:
36
IC50:
150
12
9
2D
3D
TSV
Host translation inhibitor nsp1
Ki:
36
IC50:
150
12
9
2D
3D
TSV
Leader protein
Ki:
55
IC50:
208
18
10
2D
3D
TSV
Metabotropic glutamate receptor 3 (mGlu3)
Ki:
18
IC50:
390
EC50:
88
21
1
2D
3D
TSV
NendoU
Ki:
36
IC50:
150
12
9
2D
3D
TSV
nsp12
Ki:
36
IC50:
150
12
9
2D
3D
TSV
nsp13
Ki:
36
IC50:
150
12
9
2D
3D
TSV
nsp14
Ki:
36
IC50:
150
12
9
2D
3D
TSV
nsp15
Ki:
36
IC50:
150
12
9
2D
3D
TSV
nsp16
Ki:
36
IC50:
150
12
9
2D
3D
TSV
ORF1ab polyprotein
Ki:
36
IC50:
150
12
9
2D
3D
TSV
p65 homolog
Ki:
55
IC50:
208
18
10
2D
3D
TSV
Papain-like proteinase
Ki:
55
IC50:
208
18
10
2D
3D
TSV
PL-PRO
Ki:
55
IC50:
208
18
10
2D
3D
TSV
PL2-PRO
Ki:
55
IC50:
208
18
10
2D
3D
TSV
Pol
Ki:
36
IC50:
150
12
9
2D
3D
TSV
pp1ab
Ki:
36
IC50:
150
12
9
2D
3D
TSV
RdRp
Ki:
36
IC50:
150
12
9
2D
3D
TSV
rep
Ki:
36
IC50:
150
12
9
2D
3D
TSV
Replicase polyprotein 1ab
Ki:
55
IC50:
208
18
10
2D
3D
TSV
RNA-directed RNA polymerase
Ki:
36
IC50:
152
13
9
2D
3D
TSV
SARS Coronavirus 3C-like Protease
Ki:
36
IC50:
150
12
9
2D
3D
TSV
SARS coronavirus main proteinase
Ki:
55
IC50:
208
18
10
2D
3D
TSV
Uridylate-specific endoribonuclease
Ki:
36
IC50:
150
12
9
2D
3D
TSV