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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
Compound
FDA Drugs
Important Compounds
Chemical Structure
Name
SMILES
Number of Data
/
Targets
Special tools
3D Structure Series
Find My Compound's Targets
Find Compounds for My Targets
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SCOP
Citation
Author
Journal/Citation
Institution
PubMed
PubChem BioAssay
US Patent
Special Data Sets
D3R
Host Guest Systems
Prot-Lig Validation Sets
Other Databases
PDB
85%
100%
Seq ID
UniProtKB/Swiss-Prot
UniProtKB/TrEMBL
PubMed
Download
All Compounds & Data
Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
Enter Data
Deposition
Contribute data
Sent Comments
Targets Binding with 449 Compounds
Target Name
Commercially
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Compounds
Protein/Small Molecule
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AffyNet
Ki
IC50
Kd
EC50
k
off
k
on
other
ITC
SDF
TSV
1
ALXR, FPRL1, FPR2
181
345
350
1
139
0
0
0
0
0
11
3
2D
3D
TSV
2
Endothelial nitric-oxide synthase (eNOS)
22
398
112
6
3
0
0
0
0
0
50
1
2D
3D
TSV
3
FMLP-R-I
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
4
FMLP-related receptor I
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
5
FMLP-related receptor I FMLP-R-I
181
345
350
1
139
0
0
0
0
0
11
3
2D
3D
TSV
6
Formyl peptide receptor related sequence 1
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
7
Formyl peptide receptor-like 1
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
8
Formyl peptide receptor-related sequence 1
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
9
Fpr-s1
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
10
Fpr2
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
11
Fpr3
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
12
Fprl1
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
13
hFPRL
181
345
350
1
139
0
0
0
0
0
11
3
2D
3D
TSV
14
HM63
181
345
350
1
139
0
0
0
0
0
11
3
2D
3D
TSV
15
Lipoxin A4 receptor
181
345
350
2
152
0
0
0
0
0
11
5
2D
3D
TSV
16
Lipoxin A4 receptor (LXA4)
181
345
350
1
139
0
0
0
0
0
11
3
2D
3D
TSV
17
LXA4 receptor
181
345
350
2
152
0
0
0
0
0
11
5
2D
3D
TSV
18
Lxa4r
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
19
N-formyl peptide receptor 2
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
20
N-formyl peptide receptor 3
2
0
0
1
13
0
0
0
0
0
2
3
2D
3D
TSV
21
Nitric Oxide Synthase, endothelial Mutant (N368D)
0
3
0
0
0
0
0
0
0
0
1
0
2D
3D
TSV
22
PGI receptor
41
285
173
0
76
0
0
0
0
0
63
1
2D
3D
TSV
23
Prostacyclin (IP) Receptor
41
285
173
0
76
0
0
0
0
0
63
1
2D
3D
TSV
24
Prostaglandin I2 receptor
41
285
173
0
76
0
0
0
0
0
63
1
2D
3D
TSV
25
Prostanoid IP receptor
41
285
173
0
76
0
0
0
0
0
63
1
2D
3D
TSV
26
RFP
181
345
350
1
139
0
0
0
0
0
11
3
2D
3D
TSV
27
signal transducer and activator of transcription 1 isoform alpha
281
10
305
4
135
0
0
0
0
0
15
10
2D
3D
TSV
28
Signal transducer and activator of transcription 1-alpha/beta
281
10
305
4
135
0
0
0
0
0
15
10
2D
3D
TSV
29
Transcription factor ISGF-3 components p91/p84
281
10
305
4
135
0
0
0
0
0
15
10
2D
3D
TSV
30
Transcription Factor STAT1
281
10
305
4
135
0
0
0
0
0
15
10
2D
3D
TSV
31
Transitional endoplasmic reticulum ATPase
53
0
504
0
3
0
0
0
0
0
10
14
2D
3D
TSV
32
Valosin containing protein, p97 subunit
53
0
504
0
3
0
0
0
0
0
10
14
2D
3D
TSV
33
Valosin-containing protein
53
0
504
0
3
0
0
0
0
0
10
14
2D
3D
TSV
34
Valosin-containing protein (VCP)
53
0
504
0
3
0
0
0
0
0
10
14
2D
3D
TSV
Sub total
2994
4341
6840
44
2153
0
0
0
0
0
Total
13378