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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
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Source Organism
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/
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Seq ID
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Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Targets Binding with 46 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
HDAC4 (aa 2-1084)
IC50:
46
1
0
2D
3D
TSV
Activating signal cointegrator 1 complex subunit 3-like 1
IC50:
16
3
8
2D
3D
TSV
Adrenaline alpha1
Ki:
50
IC50:
36
18
4
2D
3D
TSV
Beta-mannosidase
Ki:
35
IC50:
11
7
6
2D
3D
TSV
BRR2 homolog
IC50:
16
3
8
2D
3D
TSV
Carboxylesterase 3 precursor
IC50:
46
1
1
2D
3D
TSV
cPLA2-beta
IC50:
67
1
9
2D
3D
TSV
Cytosolic phospholipase A2 beta
IC50:
67
1
9
2D
3D
TSV
Enoyl-ACP Reductase (FabK)
IC50:
61
4
1
2D
3D
TSV
FabK
IC50:
61
4
1
2D
3D
TSV
Glutamate receptor, ionotropic kainate 5
Ki:
47
EC50:
3
7
3
2D
3D
TSV
Glutamate-Kainate 5
Ki:
47
EC50:
3
7
3
2D
3D
TSV
Glutaminyl-peptide cyclotransferase-like protein (QC)
Ki:
38
IC50:
46
3
4
2D
3D
TSV
Glyceraldehyde-3-phosphate dehydrogenase, glycosomal
Ki:
18
IC50:
39
3
1
2D
3D
TSV
Grik5
Ki:
47
EC50:
3
7
3
2D
3D
TSV
h12
IC50:
45
Kd:
3
2
7
2D
3D
TSV
Histone Deacetylase 4 (HDAC4) Mutant (H976Y)
IC50:
32
Other:
16
3
0
2D
3D
TSV
Histone deacetylase 4 gain of function (GOF) mutant
IC50:
32
Other:
16
3
0
2D
3D
TSV
NADH-dependent, FAD-containing enoyl-ACP
IC50:
61
4
1
2D
3D
TSV
Peptidase 1 (Der p 1)
IC50:
49
2
3
2D
3D
TSV
Phospholipase A2 group 1VB
IC50:
67
1
9
2D
3D
TSV
Phospholipase A2 group IVB
IC50:
67
1
9
2D
3D
TSV
Rho cDNA clone 12
IC50:
45
Kd:
3
2
7
2D
3D
TSV
rOCT1
Ki:
50
IC50:
36
18
4
2D
3D
TSV
TGH
IC50:
46
1
1
2D
3D
TSV
trans-2-enoyl-ACP reductase II
IC50:
61
4
1
2D
3D
TSV
Transforming protein RhoA
IC50:
45
Kd:
3
2
7
2D
3D
TSV
Triacylglycerol Hydrolase
IC50:
46
1
1
2D
3D
TSV
U5 small nuclear ribonucleoprotein 200 kDa helicase
IC50:
16
3
8
2D
3D
TSV
U5 snRNP-specific 200 kDa protein
IC50:
16
3
8
2D
3D
TSV
U5-200KD
IC50:
16
3
8
2D
3D
TSV
Ubiquitin carboxyl-terminal hydrolase isozyme L3 (UCH-L3)
IC50:
24
1
3
2D
3D
TSV
Ubiquitin thioesterase L3
Ki:
1
IC50:
45
Other:
2
4
7
2D
3D
TSV
UCH-L3
IC50:
24
1
3
2D
3D
TSV