Target Name | Commercially Available Compounds | Protein/Small Molecule | Other |
Articles | UniProtKB/ Swiss-Prot/TrEMBL | Download | myBDB | AffyNet |
Ki | IC50 | Kd | EC50 | koff | kon | other | ITC | SDF | TSV |
1 |
p110 alpha |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
2 |
P42336 |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
3 |
Phosphatidylinositol 3-kinase alpha (PI3Kalpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
4 |
Phosphatidylinositol 4,5-biphosphate 3-kinase catalytic subunit alpha (PIK3CA) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
5 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit (PI3K-alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
6 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha (PI3Kalpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
7 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
8 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform ( PI3K-alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
9 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (p110alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
10 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3-Ka) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
11 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K p110alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
12 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
13 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K-alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
14 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3Ka) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
15 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3Kalpha p110alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
16 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PIK3CA) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
17 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
18 |
Phosphoinositide 3-Kinase (PI3K), alpha Chain A |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
19 |
Phosphoinositide 3-kinase alpha (PI3K-alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
20 |
Phosphoinositide-3-kinase (PI3K alpha) |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
21 |
PI3-kinase subunit alpha |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
22 |
PI3-kinase subunit p110-alpha |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
23 |
PIK3CA |
184
|
1094
|
4451
|
814
|
53
|
0
|
0
|
0
|
0
|
0
|
241
|
4 |
2D 3D | TSV
|
| |
Sub total | 4232 | 25162 | 102373 | 18722 | 1219 | 0 | 0 | 0 | 0 | 0 | | | |
Total | 147476 |
---|