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Targets Binding with 5082 Compounds


Target NameCommercially
Available
Compounds
Protein/Small MoleculeOther

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AffyNet
KiIC50KdEC50koffkonotherITCSDFTSV
1 p110 alphaBDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
2 P42336BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
3 Phosphatidylinositol 3-kinase alpha (PI3Kalpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
4 Phosphatidylinositol 4,5-biphosphate 3-kinase catalytic subunit alpha (PIK3CA)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
5 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit (PI3K-alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
6 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha (PI3Kalpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
7 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformBDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
8 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform ( PI3K-alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
9 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (p110alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
10 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3-Ka)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
11 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K p110alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
12 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
13 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K-alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
14 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3Ka)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
15 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3Kalpha p110alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
16 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PIK3CA)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
17 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrialBDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
18 Phosphoinositide 3-Kinase (PI3K), alpha Chain ABDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
19 Phosphoinositide 3-kinase alpha (PI3K-alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
20 Phosphoinositide-3-kinase (PI3K alpha)BDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
21 PI3-kinase subunit alphaBDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
22 PI3-kinase subunit p110-alphaBDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
23 PIK3CABDB 184 1094 4451 814 53 0 0 0 0 0 241 4 2D 3DTSV
Sub total42322516210237318722121900000
Total147476