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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
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/
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Ki
IC50
Kd
EC50
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ΔH°
-TΔS°
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Targets Binding with 65 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
2-OG-Dependent Histone Demethylase JMJD2E
Ki:
5
IC50:
69
10
1
2D
3D
TSV
5-enolpyruvy-shikimate-3-phosphate synthase
Ki:
30
IC50:
44
Kd:
17
Koff:
3
Kon:
4
8
4
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 5
IC50:
57
Other:
8
2
0
2D
3D
TSV
ADAM-TS 11
IC50:
57
Other:
8
2
0
2D
3D
TSV
ADAMTS-5 (Aggrecanase-2)
IC50:
57
Other:
8
2
0
2D
3D
TSV
ADMP-2
IC50:
57
Other:
8
2
0
2D
3D
TSV
Bromodomain-containing protein 2 Bromo 1 domain(BRD2 BD1)
Ki:
27
IC50:
37
Kd:
4
2
0
2D
3D
TSV
Catechol O-methyltransferase
Ki:
32
IC50:
50
Kd:
4
7
9
2D
3D
TSV
Catechol O-methyltransferase (MB-COMT)
Ki:
22
IC50:
43
Kd:
4
5
6
2D
3D
TSV
Cyclic nucleotide specific phosphodiesterase
IC50:
65
2
1
2D
3D
TSV
G-protein coupled receptor 4 (GPR4)
IC50:
44
2
5
2D
3D
TSV
Histone Lysine Demethylase
Ki:
5
IC50:
69
10
1
2D
3D
TSV
Jumonji domain-containing protein 2E (JMJD2E)
Ki:
5
IC50:
69
10
1
2D
3D
TSV
KDM4D-like protein
Ki:
5
IC50:
69
10
1
2D
3D
TSV
Lysine-specific demethylase 4D-like
Ki:
5
IC50:
69
10
1
2D
3D
TSV
Lysine-specific demethylase 4E
Ki:
5
IC50:
69
10
1
2D
3D
TSV
Lysine-specific demethylase 4E (KDM4E)
Ki:
5
IC50:
69
10
1
2D
3D
TSV
mothers against decapentaplegic homolog 3
IC50:
66
2
14
2D
3D
TSV
Neuronal acetylcholine receptor protein alpha-2/beta-2 subunit
Ki:
47
IC50:
4
9
4
2D
3D
TSV
Neuronal acetylcholine receptor; alpha2/beta2
Ki:
88
IC50:
4
14
9
2D
3D
TSV
Neuronal acetylcholine recetpor; alpha2/beta2
Ki:
3
IC50:
3
3
2
2D
3D
TSV
Phosphodiesterase (TcrPDEC)
IC50:
65
2
1
2D
3D
TSV
Sialidase
Ki:
54
IC50:
85
6
5
2D
3D
TSV