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Targets Binding with 690 Compounds


Target NameCommercially
Available
Compounds
Protein/Small MoleculeOther

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AffyNet
KiIC50KdEC50koffkonotherITCSDFTSV
1 12 kDa FKBPBDB 95 400 182 107 61 0 0 0 0 0 44 11 2D 3DTSV
2 CK2- alphaBDB 3 130 674 128 0 0 0 0 0 0 48 9 2D 3DTSV
3 FK506-binding protein 1ABDB 95 400 182 107 61 0 0 0 0 0 44 11 2D 3DTSV
4 FK506-binding protein 1A (FKBP12)BDB 95 350 182 107 61 0 0 0 0 0 43 9 2D 3DTSV
5 FKBP-12BDB 95 400 182 107 61 0 0 0 0 0 44 11 2D 3DTSV
6 FKBP-1ABDB 95 350 182 107 61 0 0 0 0 0 43 9 2D 3DTSV
7 FKBP12BDB 95 350 182 107 61 0 0 0 0 0 43 9 2D 3DTSV
8 Gastric receptor IBDB 68 338 122 189 214 0 0 0 0 0 146 7 2D 3DTSV
9 H2RBDB 68 338 122 189 214 0 0 0 0 0 146 7 2D 3DTSV
10 HISTAMINE H2BDB 69 342 122 189 214 0 0 0 0 0 150 10 2D 3DTSV
11 Histamine H2 ReceptorBDB 41 244 85 0 83 0 0 0 0 0 103 5 2D 3DTSV
12 Nuclear receptor subfamily 2 group B member 1EBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
13 Peptidyl-prolyl cis-trans isomerase (FKBP)BDB 95 350 182 107 61 0 0 0 0 0 43 9 2D 3DTSV
14 Peptidyl-prolyl cis-trans isomerase FKBP1ABDB 95 350 182 107 61 0 0 0 0 0 43 9 2D 3DTSV
15 PPIase FKBP1ABDB 95 350 182 107 61 0 0 0 0 0 43 9 2D 3DTSV
16 Prolyl endopeptidaseBDB 9 105 788 0 0 3 3 0 0 0 51 9 2D 3DTSV
17 Retinoic acid receptor RXR-alphaEBI 23 191 248 128 417 0 0 0 0 0 68 6 2D 3DTSV
18 Retinoid X receptor alpha (F313A)EBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
19 Retinoid X receptor alpha (F313I)EBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
20 Retinoid X receptor alpha (F313S)EBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
21 Retinoid X receptor alpha (L436F)EBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
22 Retinoid X receptor alpha (L436V)EBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
23 Retinoid X receptor betaEBI 15 141 18 65 159 0 0 0 0 0 25 9 2D 3DTSV
24 RXR alpha/PPAR gammaEBI 22 173 231 128 403 0 0 0 0 0 65 5 2D 3DTSV
Sub total1305634054342747467100000
Total19192