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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
Chemical Structure
Pathways
Source Organism
Number of Compounds
Monomer List in csv
Het List in SDF
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Important Compounds
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Name
SMILES
Number of Data
/
Targets
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85%
100%
Seq ID
UniProtKB/Swiss-Prot
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Targets Binding with 96 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
Dual specificity mitogen-activated protein kinase kinase 3
IC50:
15
Kd:
121
12
7
2D
3D
TSV
G-protein coupled receptor 10 (GPR10)
Ki:
96
IC50:
49
2
5
2D
3D
TSV
GPR10
Ki:
96
IC50:
49
2
5
2D
3D
TSV
GST-Fibroblast growth factor receptor 3 (FGFR-3)
IC50:
96
1
1
2D
3D
TSV
KIAA1901
Ki:
1
IC50:
16
Kd:
120
12
10
2D
3D
TSV
Luciferin 4-monooxygenase
IC50:
172
2
5
2D
3D
TSV
MAP kinase kinase 3
IC50:
15
Kd:
121
12
7
2D
3D
TSV
MAPK/ERK kinase 3
IC50:
15
Kd:
121
12
7
2D
3D
TSV
MAPK/ERK kinase 3 (MEK3)
IC50:
15
Kd:
121
12
7
2D
3D
TSV
MAPKK 3
IC50:
15
Kd:
121
12
7
2D
3D
TSV
MARK1
IC50:
14
Kd:
127
14
9
2D
3D
TSV
MEK3
IC50:
15
Kd:
121
12
7
2D
3D
TSV
NEK1
Ki:
1
IC50:
16
Kd:
120
12
10
2D
3D
TSV
Never in mitosis A-related kinase 1
Ki:
1
IC50:
16
Kd:
120
12
10
2D
3D
TSV
NimA-related protein kinase 1
Ki:
1
IC50:
16
Kd:
120
12
10
2D
3D
TSV
Prolactin Releasing Peptide Receptor
Ki:
96
IC50:
49
2
5
2D
3D
TSV
Prolactin-releasing peptide receptor
Ki:
96
IC50:
49
2
5
2D
3D
TSV
Renal carcinoma antigen NY-REN-55
Ki:
1
IC50:
16
Kd:
120
12
10
2D
3D
TSV
Serine/threonine-protein kinase MARK1
IC50:
14
Kd:
127
14
9
2D
3D
TSV
Serine/threonine-protein kinase Nek1
Ki:
1
IC50:
16
Kd:
120
12
10
2D
3D
TSV