The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 27172398 |
20 |
An Unusual Natural Product Primary Sulfonamide: Synthesis, Carbonic Anhydrase Inhibition, and Protein X-ray Structures of Psammaplin C. |
Griffith University |
| 26498394 |
105 |
Inhibition of mammalian carbonic anhydrase isoforms I-XIV with a series of phenolic acid esters. |
Universit£ |
| 26347950 |
32 |
Phosphate Chemical Probes Designed for Location Specific Inhibition of Intracellular Carbonic Anhydrases. |
Griffith University |
| 25468040 |
77 |
Inhibition studies of new ureido-substituted sulfonamides incorporating a GABA moiety against human carbonic anhydrase isoforms I-XIV. |
TBA |
| 25358084 |
143 |
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX. |
Vilnius University |
| 25245672 |
5 |
Substituted thieno[2,3-b]thiophenes and related congeners: Synthesis,ß-glucuronidase inhibition activity, crystal structure, and POM analyses. |
King Saud University |
| 24689792 |
54 |
Cyclic secondary sulfonamides: unusually good inhibitors of cancer-related carbonic anhydrase enzymes. |
Griffith University |
| 23010455 |
108 |
Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases. |
Universidad Nacional De La Plata |
| 23067387 |
105 |
Tricyclic sulfonamides incorporating benzothiopyrano[4,3-c]pyrazole and pyridothiopyrano[4,3-c]pyrazole effectively inhibita- andß-carbonic anhydrase: X-ray crystallography and solution investigations on 15 isoforms. |
Universit£ |
| 22487176 |
109 |
Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins. |
Universit£ |
| 21211980 |
47 |
Characterization and anions inhibition studies of ana-carbonic anhydrase from the teleost fish Dicentrarchus labrax. |
Ondokuz Mayis University |
| 20674354 |
79 |
Carbonic anhydrase inhibitors. Antioxidant polyphenols effectively inhibit mammalian isoforms I-XV. |
Universit£ |
| 20605094 |
91 |
Carbonic anhydrase inhibitors. The X-ray crystal structure of human isoform II in adduct with an adamantyl analogue of acetazolamide resides in a less utilized binding pocket than most hydrophobic inhibitors. |
University Of Florida |
| 20472429 |
80 |
Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
| 20185318 |
132 |
Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I-XIV with a series of natural product polyphenols and phenolic acids. |
Universit£ |
| 19911821 |
273 |
Deciphering the mechanism of carbonic anhydrase inhibition with coumarins and thiocoumarins. |
Universita Degli Studi Di Firenze |
| 20028100 |
78 |
The coumarin-binding site in carbonic anhydrase accommodates structurally diverse inhibitors: the antiepileptic lacosamide as an example and lead molecule for novel classes of carbonic anhydrase inhibitors. |
Universit£ |
| 19186056 |
60 |
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases. |
Universit£ |
| 18990571 |
65 |
Carbonic anhydrase inhibitors: 2-substituted-1,3,4-thiadiazole-5-sulfamides act as powerful and selective inhibitors of the mitochondrial isozymes VA and VB over the cytosolic and membrane-associated carbonic anhydrases I, II and IV. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
| 18644716 |
52 |
Inhibition of human mitochondrial carbonic anhydrases VA and VB with para-(4-phenyltriazole-1-yl)-benzenesulfonamide derivatives. |
Griffith University |
| 18359629 |
84 |
Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
| 17475500 |
130 |
Carbonic anhydrases as targets for medicinal chemistry. |
Universit£ |
| 17420132 |
4 |
Molecular modeling study for the binding of zonisamide and topiramate to the human mitochondrial carbonic anhydrase isoform VA. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
| 17376683 |
63 |
Carbonic anhydrase inhibitors. Inhibition of isoforms I, II, IV, VA, VII, IX, and XIV with sulfonamides incorporating fructopyranose-thioureido tails. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
| 17314045 |
11 |
Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I. |
Universit£ |
| 17228881 |
141 |
Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors. |
Kochi Medical School |
| 16203142 |
55 |
Carbonic anhydrase inhibitors: inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides. |
Universit£ |
| 15664814 |
55 |
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
Universit£ |
| 22365761 |
144 |
New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II. |
Universit£ |
| 21821413 |
65 |
Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against humana- and bacterial/fungalß-carbonic anhydrases. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
| 21515057 |
153 |
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies. |
Universit£ |
| 21300547 |
64 |
(R)-/(S)-10-camphorsulfonyl-substituted aromatic/heterocyclic sulfonamides selectively inhibit mitochondrial over cytosolic carbonic anhydrases. |
Universit£ |
| 21251841 |
90 |
A newß-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth. |
University Of Montpellier |
| 20590092 |
273 |
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule. |
Universita Degli Studi Di Firenze |
| 19527930 |
53 |
The protein tyrosine kinase inhibitors imatinib and nilotinib strongly inhibit several mammalian alpha-carbonic anhydrase isoforms. |
University Of Tampere And Tampere University Hospital |
| 16759856 |
9 |
N-hydroxyurea--a versatile zinc binding function in the design of metalloenzyme inhibitors. |
Università |
| 15780631 |
55 |
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V and IX with complex fluorides, chlorides and cyanides. |
Università |
| 15745821 |
21 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with organic phosphates and phosphonates. |
University Of Montpellier |
| 15664815 |
45 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with carboxylates. |
Università |
| 15482952 |
48 |
Carbonic anhydrase inhibitors: inhibition of human cytosolic isozyme II and mitochondrial isozyme V with a series of benzene sulfonamide derivatives. |
Università |
| 12065583 |
3 |
Identification of a novel human eicosanoid receptor coupled to G(i/o). |
Tanabe Seiyaku |
| 10945872 |
14 |
Pharmacological actions of a novel, high-affinity, and selective human dopamine D(3) receptor antagonist, SB-277011-A. |
Smithkline Beecham Pharmaceuticals |
| 7815325 |
65 |
Cloning and pharmacological characterization of human alpha-1 adrenergic receptors: sequence corrections and direct comparison with other species homologues. |
Duke University |
| 3130534 |
3 |
7-[3-(4-[2,3-Dimethylphenyl]piperazinyl)propoxy]-2(1H)-quinolinone (OPC-4392), a presynaptic dopamine autoreceptor agonist and postsynaptic D2 receptor antagonist. |
Tokushima Research Institute |
| 2664084 |
17 |
Detection of a novel serotonin receptor subtype (5-HT1E) in human brain: interaction with a GTP-binding protein. |
Albany Medical College |
| 2547939 |
11 |
Characterization of the striatal M2 muscarinic receptor mediating inhibition of cyclic AMP using selective antagonists: a comparison with the brainstem M2 receptor. |
Abbott Laboratories |
| 2537406 |
2 |
Pharmacological characterization of the M1 muscarinic receptors expressed in murine fibroblast B82 cells. |
University Of Arizona |
| 19900813 |
12 |
Optimization of (4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepine-5-ylidene)acetamide derivatives as arginine vasopressin V2 receptor agonists and discussion of their binding modes. |
Astellas Pharma |
| 19102698 |
16 |
Discovery of 1-[9-(4-chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxylic acid amide hydrochloride (CP-945,598), a novel, potent, and selective cannabinoid type 1 receptor antagonist. |
Pfizer |
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