The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
10464022 |
25 |
Design and in vivo analysis of potent non-thiol inhibitors of farnesyl protein transferase. |
Merck Research Laboratories |
9784104 |
30 |
Potent and selective non-cysteine-containing inhibitors of protein farnesyltransferase. |
Abbott Laboratories |
9651171 |
29 |
N-Arylalkyl pseudopeptide inhibitors of farnesyltransferase. |
Merck Research Laboratories |
9003517 |
63 |
Structure-activity relationships of cysteine-lacking pentapeptide derivatives that inhibit ras farnesyltransferase. |
Warner-Lambert |
9301658 |
53 |
Ras farnesyltransferase: a new therapeutic target. |
Warner-Lambert |
8145221 |
28 |
Pseudopeptide inhibitors of Ras farnesyl-protein transferase. |
Merck Research Laboratories |
12668011 |
22 |
Synthesis and evaluation of a novel series of farnesyl protein transferase inhibitors as non-peptidic CAAX tetrapeptide analogues. |
Centre De Recherche Pierre Fabre |
10450988 |
51 |
Synthesis and evaluation of hydroxyproline-derived isoprenyltransferase inhibitors. |
Eisai Research Institute |
| 21 |
DIARYLETHER INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE |
TBA |
| 20 |
Inhibition of farnesyl protein transferase by new farnesyl phosphonate derivatives of phenylalanine |
TBA |
| 23 |
Local constrained shifty pseudopeptides inhibitors of rasfarnesyl transferase |
TBA |
15582430 |
123 |
Design and synthesis of o-trifluoromethylbiphenyl substituted 2-amino-nicotinonitriles as inhibitors of farnesyltransferase. |
Abbott Laboratories |
15454229 |
86 |
Synthesis and activity of 1-aryl-1'-imidazolyl methyl ethers as non-thiol farnesyltransferase inhibitors. |
Abbott Laboratories |
15454228 |
17 |
Design, synthesis, and activity of 4-quinolone and pyridone compounds as nonthiol-containing farnesyltransferase inhibitors. |
Abbott Laboratories |
15324873 |
21 |
Synthesis of 1H-pyridin-2-one derivatives as potent and selective farnesyltransferase inhibitors. |
Abbott Laboratories |
12852971 |
8 |
Improvement of biological activity and proteolytic stability of peptides by coupling with a cyclic peptide. |
Kyowa Hakko Kogyo |
12773050 |
26 |
Discovery and structure-activity relationships of novel piperidine inhibitors of farnesyltransferase. |
Pharmaceutical Research Institute |
12699757 |
72 |
Discovery of potent imidazole and cyanophenyl containing farnesyltransferase inhibitors with improved oral bioavailability. |
Abbott Laboratories |
12668012 |
15 |
From pure FPP to mixed FPP and CAAX competitive inhibitors of farnesyl protein transferase. |
Centre De Recherche Pierre Fabre |
12657284 |
31 |
Novel and selective imidazole-containing biphenyl inhibitors of protein farnesyltransferase. |
Abbott Laboratories |
12039571 |
19 |
Development of tripeptidyl farnesyltransferase inhibitors. |
Department Of Chemistry And School Of Molecular Science(Bk21) |
11965368 |
64 |
Potent inhibitors of farnesyltransferase and geranylgeranyltransferase-I. |
Merck Research Laboratories |
10612589 |
22 |
Imidazole-containing diarylether and diarylsulfone inhibitors of farnesyl-protein transferase. |
Merck Research Laboratories |
10479301 |
27 |
Second-generation peptidomimetic inhibitors of protein farnesyltransferase demonstrating improved cellular potency and significant in vivo efficacy. |
Abbott Laboratories |
8691462 |
14 |
2-substituted piperazines as constrained amino acids. Application to the synthesis of potent, non carboxylic acid inhibitors of farnesyltransferase. |
Merck Research Laboratories |
7562930 |
34 |
Pseudodipeptide inhibitors of protein farnesyltransferase. |
Merck Research Laboratories |
12816482 |
38 |
Complexation and chiral recognition thermodynamics of gamma-cyclodextrin with N-acetyl- and N-carbobenzyloxy-dipeptides possessing two aromatic rings. |
Japan Science And Technology Agency |
12657282 |
13 |
Aryl tetrahydropyridine inhibitors of farnesyltransferase: glycine, phenylalanine and histidine derivatives. |
Abbott Laboratories |
15808463 |
35 |
Design, synthesis, and activity of achiral analogs of 2-quinolones and indoles as non-thiol farnesyltransferase inhibitors. |
Abbott Laboratories |
15911281 |
30 |
Benzimidazolones and indoles as non-thiol farnesyltransferase inhibitors based on tipifarnib scaffold: synthesis and activity. |
Abbott Laboratories |