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27 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
10201825 2 Solid-phase synthesis of benzisothiazolones as serine protease inhibitors.EBI Bristol-Myers Squibb Pharmaceutical Research Institute
26122211 3 Discovery of non-competitive thrombin inhibitor derived from competitive tryptase inhibitor skeleton: Shift in molecular recognition resulted from skeletal conversion of carboxylate into phosphonate.EBI Tokyo University Of Pharmacy And Life Sciences
16644215 52 Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors.EBI Celera Genomics
16554154 9 Development of activity-based probes for trypsin-family serine proteases.EBI Celera Genomics
19715320 87 Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI University Of Florida
12930148 41 Potent, small-molecule inhibitors of human mast cell tryptase. Antiasthmatic action of a dipeptide-based transition-state analogue containing a benzothiazole ketone.EBI Johnson & Johnson Pharmaceutical Research & Development
15081015 91 Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors.EBI The Bristol-Myers Squibb Pharmaceutical Research Institute
16725321 13 Novel, potent, selective, and orally bioavailable human betaII-tryptase inhibitors.EBI Celera Genomics
16714109 40 Design of novel, potent, and selective human beta-tryptase inhibitors based on alpha-keto-[1,2,4]-oxadiazoles.EBI Celera
16540315 23 Synthesis and evaluation of 4-substituted benzylamine derivatives as beta-tryptase inhibitors.EBI Mochida Pharmaceutical
15911249 29 Design, synthesis, and biological activity of potent and selective inhibitors of mast cell tryptase.EBI Aventis Pharmaceuticals
15745817 14 Combinatorial approaches towards the discovery of new tryptase inhibitors.EBI University Of Barcelona
15546728 15 Design of bivalent ligands using hydrogen bond linkers: synthesis and evaluation of inhibitors for human beta-tryptase.EBI Aventis Pharmaceuticals
15341931 15 Novel pyrazinone inhibitors of mast cell tryptase: synthesis and SAR evaluation.EBI Aventis Pharmaceuticals
15081014 35 Synthesis of potent and highly selective nonguanidine azetidinone inhibitors of human tryptase.EBI The Bristol-Myers Squibb Pharmaceutical Research Institute
14698147 60 Synthesis of potent and selective 2-azepanone inhibitors of human tryptase.EBI The Bristol-Myers Squibb Pharmaceutical Research Institute
11959009 7 Bivalent inhibition of beta-tryptase: distance scan of neighboring subunits by dibasic inhibitors.EBI Institut FüR Biochemie
11527724 30 Monocharged inhibitors of mast cell tryptase derived from potent and selective dibasic inhibitors.EBI Axys Pharmaceuticals
11425524 62 Dibasic inhibitors of human mast cell tryptase. Part 3: identification of a series of potent and selective inhibitors containing the benzamidine functionality.EBI Axys Pharmaceuticals
11055356 236 Dibasic inhibitors of human mast cell tryptase. Part 2: structure-activity relationships and requirements for potent activity.EBI Axys Pharmaceuticals
11055355 72 Dibasic inhibitors of human mast cell tryptase. Part 1: synthesis and optimization of a novel class of inhibitors.EBI Axys Pharmaceuticals
10612586 34 Syntheses and evaluation of amidinobenzofuran derivatives as tryptase inhibitors.EBI Yoshitomi Pharmaceutical Industries
9873535 13 Highly efficient and versatile synthesis of libraries of constrained beta-strand mimetics.EBI Molecumetics