The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
1507209 |
7 |
Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative structure-activity relationships of substituted 4- and 5-(2-aminoethyl)thiazoles. |
Vrije Universiteit |
20409707 |
66 |
Chiral NG-acylated hetarylpropylguanidine-type histamine H2 receptor agonists do not show significant stereoselectivity. |
University Of Regensburg |
19317445 |
53 |
N(G)-acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent. |
University Of Regensburg |
18976927 |
83 |
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. |
Universit£ |
9548813 |
53 |
The selective 5-HT1B receptor inverse agonist 1'-methyl-5-[[2'-methyl-4'-(5-methyl-1,2, 4-oxadiazol-3-yl)biphenyl-4-yl]carbonyl]-2,3,6,7-tetrahydro- spiro[furo[2,3-f]indole-3,4'-piperidine] (SB-224289) potently blocks terminal 5-HT autoreceptor function both in vitro and in vivo. |
Smithkline Beecham Pharmaceuticals |
1613748 |
8 |
Iodoaminopotentidine and related compounds: a new class of ligands with high affinity and selectivity for the histamine H2 receptor. |
Freie Universit£T Berlin |
2931524 |
19 |
The histamine H2 receptor agonist impromidine: synthesis and structure-activity considerations. |
TBA |
6131129 |
10 |
Conformational requirements for histamine H2-receptor inhibitors: a structure-activity study of phenylene analogues related to cimetidine and tiotidine. |
TBA |
6121913 |
5 |
Inhibitors of gastric acid secretion: 3,4-diamino-1,2,5-thiadiazole 1-oxides and 1,1-dioxides as urea equivalents in a series of histamine H2-receptor antagonists. |
TBA |
22216892 |
66 |
The bivalent ligand approach leads to highly potent and selective acylguanidine-type histamine H2 receptor agonists. |
University Of Regensburg |
20875743 |
90 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: design, synthesis, and structure-activity rela |
Pfizer |
18950149 |
75 |
Acylguanidines as bioisosteres of guanidines: NG-acylated imidazolylpropylguanidines, a new class of histamine H2 receptor agonists. |
University Of Regensburg |
12672253 |
60 |
Novel nonimidazole histamine H3 receptor antagonists: 1-(4-(phenoxymethyl)benzyl)piperidines and related compounds. |
Freie Universit£T Berlin |
12190321 |
55 |
Influence of bulky substituents on histamine h(3) receptor agonist/antagonist properties. |
Freie Universit£T Berlin |
10447960 |
20 |
Development of predictive retention-activity relationship models of tricyclic antidepressants by micellar liquid chromatography. |
Universidad De Valencia |
7904648 |
3 |
Studies on antiulcer drugs. 7. 2-Guanidino-4-pyridylthiazoles as histamine H2-receptor antagonists with potent gastroprotective effects against nonsteroidal antiinflammatory drug-induced injury. |
Fujisawa Pharmaceutical |
20812727 |
157 |
Synthesis, structure-affinity relationships, and radiolabeling of selective high-affinity 5-HT4 receptor ligands as prospective imaging probes for positron emission tomography. |
National Institute Of Mental Health |
16730977 |
2 |
Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine. |
The University Of Kansas |
15115409 |
72 |
4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists. |
Freie UniversitäT Berlin |
11855993 |
91 |
Development of a new class of nonimidazole histamine H(3) receptor ligands with combined inhibitory histamine N-methyltransferase activity. |
Freie UniversitäT Berlin |
10966752 |
60 |
New histamine H(3)-receptor ligands of the proxifan series: imoproxifan and other selective antagonists with high oral in vivo potency. |
Freie UniversitäT Berlin |
8676353 |
140 |
Novel carbamates as potent histamine H3 receptor antagonists with high in vitro and oral in vivo activity. |
Freie UniversitäT Berlin |
6192241 |
15 |
Synthesis and biological properties of thiophene ring analogues of mianserin. |
TBA |