The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27287367 |
36 |
Evaluation of bisbenzamidines as inhibitors for matriptase-2. |
University Of Bonn |
26421993 |
44 |
Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors. |
Aurigene Discovery Technologies |
24794746 |
168 |
Structure-guided discovery of 1,3,5 tri-substituted benzenes as potent and selective matriptase inhibitors exhibiting in vivo antitumor efficacy. |
Aurigene Discovery Technologies |
20503967 |
138 |
Factor Xa inhibitors: next-generation antithrombotic agents. |
Bristol-Myers Squibb |
10956211 |
14 |
GRID/CPCA: a new computational tool to design selective ligands. |
Boehringer Ingelheim Pharma |
9301673 |
234 |
Synthesis and structure-activity relationships of potent thrombin inhibitors: piperazides of 3-amidinophenylalanine. |
Klinikum Der Friedrich-Schiller-Universit£T Jena |
10498204 |
25 |
Aminoisoquinolines: design and synthesis of an orally active benzamidine isostere for the inhibition of factor XA. |
Rh£Ne-Poulenc Rorer |
19805567 |
3 |
Long-lasting enfuvirtide carrier pentasaccharide conjugates with potent anti-human immunodeficiency virus type 1 activity. |
Endotis Pharma |
| 32 |
Bisbenzamidine isoxazoline derivatives as factor Xa inhibitors |
TBA |
| 13 |
Characterization of LY806303 as a potent and selective inhibitor of thrombin |
TBA |
16970403 |
74 |
Diphenyl phosphonate inhibitors for the urokinase-type plasminogen activator: optimization of the P4 position. |
University Of Antwerp |
12036353 |
38 |
Design of selective thrombin inhibitors based on the (R)-Phe-Pro-Arg sequence. |
Pfizer |
10636232 |
58 |
Design, synthesis and structure-activity relationship of a series of arginine aldehyde factor Xa inhibitors. Part 1: structures based on the (D)-Arg-Gly-Arg tripeptide sequence. |
Cor Therapeutics |
10560742 |
85 |
3-Amidinophenylalanine-based inhibitors of urokinase. |
UniversitäT Jena |
9876114 |
111 |
Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: implications for the inhibition of factor Xa, tPA, and urokinase. |
Institut FüR Biochemie |
9784099 |
84 |
Design of benzamidine-type inhibitors of factor Xa. |
Institut FüR Biochemie |
7473571 |
90 |
Structure-activity study of tripeptide thrombin inhibitors using alpha-alkyl amino acids and other conformationally constrained amino acid substitutions. |
Eli Lilly |