The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
23218714 |
14 |
Development of an in vivo active, dual EP1 and EP3 selective antagonist based on a novel acyl sulfonamide bioisostere. |
Vanderbilt University School Of Medicine |
22546206 |
162 |
Synthesis and evaluation of¿-lactam analogs of PGE2 as EP4 and EP2/EP4 agonists. |
Minase Research Institute |
15357992 |
81 |
Discovery of new chemical leads for prostaglandin D2 receptor antagonists. |
Minase Research Institute |
22386979 |
104 |
Discovery of novel prostaglandin analogs as potent and selective EP2/EP4 dual agonists. |
Minase Research Institute |
22119471 |
64 |
Discovery of a novel EP2/EP4 dual agonist with high subtype-selectivity. |
Minase Research Institute |
22204740 |
135 |
Synthesis and evaluation of novel modified¿-lactam prostanoids as EP4 subtype-selective agonists. |
Minase Research Institute |
21885288 |
109 |
Design and synthesis of new prostaglandin D2 receptor antagonists. |
Minase Research Institute |
21737285 |
138 |
Discovery of selective indole-based prostaglandin D2 receptor antagonist. |
Minase Research Institute |
20385498 |
115 |
3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 3: Synthesis, metabolic stability, and biological evaluation of optically active analogs. |
Minase Research Institute |
20346663 |
76 |
Discovery of novel N-acylsulfonamide analogs as potent and selective EP3 receptor antagonists. |
Minase Research Institute |
20004584 |
57 |
3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. Part 1: discovery and exploration of the carboxyamide side chain. |
Minase Research Institute |
20129791 |
120 |
3-(2-Aminocarbonylphenyl)propanoic acid analogs as potent and selective EP3 receptor antagonists. part 2: optimization of the side chains to improve in vitro and in vivo potencies. |
Minase Research Institute |
15341946 |
92 |
Discovery of orally active prostaglandin D2 receptor antagonists. |
Minase Research Institute |
11454474 |
84 |
Design and synthesis of a highly selective EP4-receptor agonist. Part 2: 5-thia and 9beta-haloPG derivatives with improved stability. |
Minase Research Institute |
11454473 |
119 |
Design and synthesis of a highly selective EP4-receptor agonist. Part 1: 3,7-dithiaPG derivatives with high selectivity. |
Minase Research Institute |
11454472 |
107 |
Design and synthesis of a highly selective EP2-receptor agonist. |
Minase Research Institute |
12192085 |
52 |
Salvinorin A: a potent naturally occurring nonnitrogenous kappa opioid selective agonist. |
Case Western Reserve University |