The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 26296911 |
11 |
3-Benzamides and 3,4,5-trimethoxyphenyl amines as calcium channel blockers. |
Ewha Womans University |
| 24936234 |
42 |
Synthesis and biological evaluation of a selective N- and p/q-type calcium channel agonist. |
TBA |
| 23098566 |
17 |
Aminopiperidine sulfonamide Cav2.2 channel inhibitors for the treatment of chronic pain. |
Merck Research Laboratories |
| 22560585 |
16 |
Discovery and evaluation of selective N-type calcium channel blockers: 6-unsubstituted-1,4-dihydropyridine-5-carboxylic acid derivatives. |
Ajinomoto Pharmaceuticals |
| 17483457 |
58 |
A-803467, a potent and selective Nav1.8 sodium channel blocker, attenuates neuropathic and inflammatory pain in the rat. |
Abbott Laboratories |
| 15537361 |
9 |
Design, synthesis, and preliminary pharmacological evaluation of 4-aminopiperidine derivatives as N-type calcium channel blockers active on pain and neuropathic pain. |
Universit£ |
| 11000000 |
1 |
(S)-4-Methyl-2-(methylamino)pentanoic acid [4, 4-bis(4-fluorophenyl)butyl]amide hydrochloride, a novel calcium channel antagonist, is efficacious in several animal models of pain. |
Pfizer |
| 22177784 |
2 |
In vivo evaluation of oral anti-tumoral effect of 3,4-dihydroquinazoline derivative on solid tumor. |
Kyung Hee University |
| 21316226 |
12 |
Pyridyl amides as potent inhibitors of T-type calcium channels. |
Merck Research Laboratories |
| 21195616 |
26 |
A potent and selective indole N-type calcium channel (Ca(v)2.2) blocker for the treatment of pain. |
Merck Research Laboratories |
| 20934333 |
2 |
Design, syntheses, and SAR of 2,8-diazaspiro[4.5]decanones as T-type calcium channel antagonists. |
Icagen |
| 20855211 |
91 |
Subtype-selective Na(v)1.8 sodium channel blockers: identification of potent, orally active nicotinamide derivatives. |
Abbott Laboratories |
| 20382529 |
13 |
Synthesis and biological evaluation of 1,4-diazepane derivatives as T-type calcium channel blockers. |
Institute Of Science And Technology |
| 17134896 |
41 |
Synthesis and SAR of novel 2-arylthiazolidinones as selective analgesic N-type calcium channel blockers. |
Ionix Pharmaceuticals |
| 16722655 |
28 |
Discovery of a novel, orally active, small molecule gonadotropin-releasing hormone (GnRH) receptor antagonist. |
Pfizer |
| 12161113 |
8 |
L-Cysteine based N-type calcium channel blockers: structure-activity relationships of the C-terminal lipophilic moiety, and oral analgesic efficacy in rat pain models. |
Minase Research Institute |
| 11958993 |
23 |
Structure-activity study of L-cysteine-based N-type calcium channel blockers: optimization of N- and C-terminal substituents. |
Minase Research Institute |
| 11514140 |
17 |
Structure-activity study and analgesic efficacy of amino acid derivatives as N-type calcium channel blockers. |
No Pharmaceutical |
| 10714496 |
4 |
Design and biological evaluation of non-peptide analogues of omega-conotoxin MVIIA. |
Parke-Davis Neuroscience Research Centre |
| 10514294 |
15 |
Synthesis of a series of 4-benzyloxyaniline analogues as neuronal N-type calcium channel blockers with improved anticonvulsant and analgesic properties. |
Warner-Lambert |
| 10476886 |
14 |
Structure-activity relationship at the proximal phenyl group in a series of non-peptidyl N-type calcium channel antagonists. |
Parke-Davis Pharmaceutical Research |
| 10476885 |
14 |
Synthesis and biological activity of substituted bis-(4-hydroxyphenyl)methanes as N-type calcium channel blockers. |
Warner-Lambert |
| 10465535 |
14 |
Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers. |
Warner-Lambert |
| 10406647 |
30 |
Multiple parallel synthesis of N,N-dialkyldipeptidylamines as N-type calcium channel blockers. |
Warner-Lambert |
| 10328297 |
13 |
Synthesis and biological evaluation of substituted 4-(OBz)phenylalanine derivatives as novel N-type calcium channel blockers. |
Warner-Lambert |
| 10206559 |
18 |
N,N-dialkyl-dipeptidylamines as novel N-type calcium channel blockers. |
Warner-Lambert |
| 9873552 |
12 |
Synthesis and structure-activity relationship of substituted 1,2,3,4-tetrahydroisoquinolines as N-type calcium channel blockers. |
Warner-Lambert |
| 26833890 |
18 |
Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease. |
Yogi Vemana University |
| 26469307 |
7 |
Phosphorylation of Capsaicinoid Derivatives Provides Highly Potent and Selective Inhibitors of the Transcription Factor STAT5b. |
University Of Leipzig |
| 12534275 |
32 |
A major role for a set of non-active site mutations in the development of HIV-1 protease drug resistance. |
The Johns Hopkins University |
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