The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 28131094 |
66 |
New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation. |
Universities Of Lille |
| 8411005 |
42 |
2-Amido-8-methoxytetralins: a series of nonindolic melatonin-like agents. |
University Of Groningen |
| 27876250 |
60 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH |
Jagiellonian University Medical College |
| 26988801 |
55 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents. |
Jagiellonian University Medical College |
| 26390077 |
42 |
Tactical Approaches to Interconverting GPCR Agonists and Antagonists. |
University Of Minnesota |
| 26820449 |
84 |
Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives. |
Universit£ |
| 26785296 |
32 |
Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity. |
Universit£ |
| 26367450 |
4 |
New coumarin-based fluorescent melatonin ligands. Design, synthesis and pharmacological characterization. |
Iqm-Csic |
| 26334942 |
43 |
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines. |
Universit£ |
| 26023814 |
79 |
Novel N-Acetyl Bioisosteres of Melatonin: Melatonergic Receptor Pharmacology, Physicochemical Studies, and Phenotypic Assessment of Their Neurogenic Potential. |
Iqm-Csic |
| 24930835 |
18 |
Synthesis of new melatoninergic hexahydroindenopyridines. |
Universidad De Valencia |
| 25232966 |
52 |
Efficient synthesis of hexahydroindenopyridines and their potential as melatoninergic ligands. |
Universidad De Valencia |
| 24228714 |
64 |
MT1 and MT2 melatonin receptors: ligands, models, oligomers, and therapeutic potential. |
The German University In Cairo |
| 23228808 |
22 |
Development of substituted N-[3-(3-methoxylphenyl)propyl] amides as MT(2)-selective melatonin agonists: improving metabolic stability. |
Hong Kong University Of Science And Technology |
| 23265885 |
30 |
Synthesis of new N-(arylcyclopropyl)acetamides and N-(arylvinyl)acetamides as conformationally-restricted ligands for melatonin receptors. |
Paris-Sud University |
| 21775151 |
22 |
Bivalent ligand approach on N-{2-[(3-methoxyphenyl)methylamino]ethyl}acetamide: synthesis, binding affinity and intrinsic activity for MT(1) and MT(2) melatonin receptors. |
Universit£ |
| 20674373 |
84 |
Design, synthesis, and pharmacological effects of structurally simple ligands for MT(1) and MT(2) melatonin receptors. |
Universit£ |
| 9804685 |
142 |
Pharmacophoric search and 3D-QSAR comparative molecular field analysis studies on agonists of melatonin sheep receptors. |
Universit£ |
| 22465637 |
48 |
4-(1-Phenyl-1H-pyrazol-4-yl)quinolines as novel, selective and brain penetrant metabotropic glutamate receptor 4 positive allosteric modulators. |
Lundbeck Research Usa |
| 21726069 |
98 |
Tryptophan 2,3-dioxygenase (TDO) inhibitors. 3-(2-(pyridyl)ethenyl)indoles as potential anticancer immunomodulators. |
University Of Namur |
| 20684563 |
176 |
Discovery of N-{1-[3-(3-oxo-2,3-dihydrobenzo[1,4]oxazin-4-yl)propyl]piperidin-4-yl}-2-phenylacetamide (Lu AE51090): an allosteric muscarinic M1 receptor agonist with unprecedented selectivity and procognitive potential. |
H. Lundbeck |
| 20444610 |
71 |
Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands. |
University Of Lille |
| 11585444 |
295 |
From hit to lead. Analyzing structure-profile relationships. |
Universities Of Lille |
| 10737738 |
78 |
Mapping the melatonin receptor. 6. Melatonin agonists and antagonists derived from 6H-isoindolo[2,1-a]indoles, 5,6-dihydroindolo[2,1-a]isoquinolines, and 6,7-dihydro-5H-benzo[c]azepino[2,1-a]indoles. |
King'S College London |
| 21764185 |
12 |
Design and synthesis of 2-phenylimidazo[1,2-a]pyridines as a novel class of melatonin receptor ligands. |
Universit£ |
| 21568291 |
30 |
Synthesis of a novel series of tricyclic dihydrofuran derivatives: discovery of 8,9-dihydrofuro[3,2-c]pyrazolo[1,5-a]pyridines as melatonin receptor (MT1/MT2) ligands. |
Takeda Pharmaceutical |
| 21392858 |
28 |
Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands. |
University Of Lille |
| 21473625 |
42 |
1,6-Dihydro-2H-indeno[5,4-b]furan derivatives: design, synthesis, and pharmacological characterization of a novel class of highly potent MT2-selective agonists. |
Takeda Pharmaceutical |
| 21377769 |
30 |
Design and synthesis of naphthalenic derivatives as new ligands at the melatonin binding site MT3. |
University Of Lille |
| 21420861 |
50 |
Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists. |
Universit£ |
| 20591666 |
66 |
A new group of oxime carbamates as reversible inhibitors of fatty acid amide hydrolase. |
Università |
| 20227878 |
40 |
Synthesis of substituted N-[3-(3-methoxyphenyl)propyl] amides as highly potent MT(2)-selective melatonin ligands. |
Hong Kong University Of Science And Technology |
| 19473848 |
7 |
Synthesis and pharmacological evaluation of 1,2,3,4-tetrahydropyrazino[1,2-a]indole and 2-[(phenylmethylamino)methyl]-1H-indole analogues as novel melatoninergic ligands. |
University Of W£Rzburg |
| | 26 |
The development of a charged melatonin receptor ligand |
TBA |
| | 12 |
Synthesis and receptor binding studies of quinolinic derivatives as melatonin receptor ligands |
TBA |
| 19193160 |
42 |
2-[(2,3-dihydro-1H-indol-1-yl)methyl]melatonin analogues: a novel class of MT2-selective melatonin receptor antagonists. |
University Of WüRzburg |
| 18778943 |
53 |
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands. |
University Of Lille 2 |
| 18657980 |
14 |
Synthesis and pharmacological evaluation of pentacyclic 6a,7-dihydrodiindole and 2,3-dihydrodiindole derivatives as novel melatoninergic ligands. |
University Of WüRzburg |
| 18372181 |
32 |
Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3. |
Université |
| 17481904 |
24 |
Synthesis and biological activity of new melatonin dimeric derivatives. |
Università |
| 16759094 |
70 |
Mapping the melatonin receptor. 7. Subtype selective ligands based on beta-substituted N-acyl-5-methoxytryptamines and beta-substituted N-acyl-5-methoxy-1-methyltryptamines. |
University Of Athens |
| 15713384 |
28 |
(R)-2-(4-Phenylbutyl)dihydrobenzofuran derivatives as melatoninergic agents. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15501061 |
51 |
Tetrahydroisoquinoline derivatives as melatonin MT2 receptor antagonists. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15380218 |
40 |
N-[2-[2-(4-Phenylbutyl)benzofuran-4-yl]cyclopropylmethyl]acetamide: an orally bioavailable melatonin receptor agonist. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15203165 |
80 |
Synthesis and structure-activity relationship of novel benzoxazole derivatives as melatonin receptor agonists. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 15013015 |
76 |
4-Substituted anilides as selective melatonin MT2 receptor agonists. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 14980664 |
48 |
Design and synthesis of benzoxazole derivatives as novel melatoninergic ligands. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 14643330 |
40 |
Heterocyclic aminopyrrolidine derivatives as melatoninergic agents. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 12646022 |
22 |
Design and synthesis of naphthalenic dimers as selective MT1 melatoninergic ligands. |
Université |
| 12643943 |
43 |
Indanyl piperazines as melatonergic MT2 selective agents. |
Bristol-Myers Squibb Pharmaceutical Research Institute |
| 12213063 |
4 |
Synthesis of a novel series of tricyclic indan derivatives as melatonin receptor agonists. |
Takeda Chemical Industries |
| 12213062 |
70 |
Synthesis of a novel series of benzocycloalkene derivatives as melatonin receptor agonists. |
Takeda Chemical Industries |
| 12061881 |
94 |
Synthesis and structure-affinity-activity relationships of novel benzofuran derivatives as MT(2) melatonin receptor selective ligands. |
Institut De Chimie Pharmaceutique Albert Lespagnol |
| 11960497 |
36 |
Synthesis of nitroindole derivatives with high affinity and selectivity for melatoninergic binding sites MT(3). |
Institut De Chimie Pharmaceutique Albert Lespagnol |
| 11063602 |
84 |
Synthesis of phenalene and acenaphthene derivatives as new conformationally restricted ligands for melatonin receptors. |
Paris-Sud University |
| 9435890 |
7 |
Development of a high-affinity ligand that binds irreversibly to Mel1b melatonin receptors. |
Duquesne University |
| 27894776 |
26 |
Design, synthesis, cyclooxygenase inhibition and biological evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing amino/methanesulfonyl pharmacophore. |
Beni-Suef University |
| 26833890 |
18 |
Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease. |
Yogi Vemana University |
| 25711384 |
19 |
Synthesis and Evaluation of 3-(furo[2,3-b]pyridin-3-yl)-4-(1H-indol-3-yl)-maleimides as Novel GSK-3ß Inhibitors and Anti-Ischemic Agents. |
Zhejiang University Of Technology |
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