The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26824643 |
69 |
Mimicking of Arginine by Functionalized N(¿)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. |
University Of Regensburg |
24900634 |
36 |
Design and Synthesis of Peptide YY Analogues with C-terminal Backbone Amide-to-Ester Modifications. |
University Of Copenhagen |
24074877 |
135 |
Dimeric argininamide-type neuropeptide Y receptor antagonists: chiral discrimination between Y1 and Y4 receptors. |
University Of Regensburg |
24090364 |
96 |
Replacement of Thr32 and Gln34 in the C-terminal neuropeptide Y fragment 25-36 by cis-cyclobutane and cis-cyclopentane β-amino acids shifts selectivity toward the Y(4) receptor. |
University Of Regensburg |
18160282 |
40 |
Discovery of novel orally active ureido NPY Y5 receptor antagonists. |
Schering-Plough Research Institute |
21782428 |
61 |
Discovery of Lu AA33810: a highly selective and potent NPY5 antagonist with in vivo efficacy in a model of mood disorder. |
Lundbeck Research Usa |
19616955 |
34 |
Discovery of pyridone-containing imidazolines as potent and selective inhibitors of neuropeptide Y Y5 receptor. |
Tsukuba Research Institute |
21493077 |
39 |
Red-fluorescent argininamide-type NPY Y1 receptor antagonists as pharmacological tools. |
Universit£T Regensburg |
19864135 |
43 |
Discovery and SAR of cyclic isothioureas as novel NPY Y1 receptor antagonists. |
Schering-Plough Research Institute |
20042335 |
12 |
[Lys(DOTA)4]BVD15, a novel and potent neuropeptide Y analog designed for Y1 receptor-targeted breast tumor imaging. |
Universit£ |
19679469 |
26 |
Identification of positron emission tomography ligands for NPY Y5 receptors in the brain. |
Tsukuba Research Institute |
19640706 |
25 |
Synthesis and evaluation of a series of 2,4-diaminopyridine derivatives as potential positron emission tomography tracers for neuropeptide Y Y1 receptors. |
Tsukuba Research Institute |
19596193 |
72 |
Design, synthesis and evaluation of a novel cyclohexanamine class of neuropeptide Y Y1 receptor antagonists. |
Tsukuba Research Institute |
19464889 |
43 |
Aryl urea derivatives of spiropiperidines as NPY Y5 receptor antagonists. |
Tsukuba Research Institute |
19459652 |
56 |
Discovery of tetrasubstituted imidazolines as potent and selective neuropeptide Y Y5 receptor antagonists: reduced human ether-a-go-go related gene potassium channel binding affinity and potent antiobesity effect. |
Tsukuba Research Institute |
19053784 |
19 |
Guanidine-acylguanidine bioisosteric approach in the design of radioligands: synthesis of a tritium-labeled N(G)-propionylargininamide ([3H]-UR-MK114) as a highly potent and selective neuropeptide Y Y1 receptor antagonist. |
University Of Regensburg |
18752943 |
36 |
Syntheses and structure-activity relationships of novel, potent, and selective trans-2-[3-oxospiro[isobenzofuran-1(3H),1'-cyclohexan]-4'-yl]benzimidazole NPY Y5 receptor antagonists. |
Banyu Tsukuba Research Institute |
18723347 |
59 |
Design, syntheses, and structure-activity relationships of novel NPY Y5 receptor antagonists: 2-{3-Oxospiro[isobenzofuran-1(3H),4'-piperidin]-1'-yl}benzimidazole derivatives. |
Banyu Tsukuba Research Institute |
18637668 |
38 |
(9S)-9-(2-hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one, a selective and orally active neuropeptide Y Y5 receptor antagonist. |
Tsukuba Research Institute |
16610810 |
39 |
Neuropeptide Y (NPY) Y4 receptor selective agonists based on NPY(32-36): development of an anorectic Y4 receptor selective agonist with picomolar affinity. |
University Of Cincinnati |
15109631 |
86 |
Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists. |
Novartis Pharma |
11334558 |
42 |
Highly selective and potent neuropeptide Y (NPY) Y1 receptor antagonists based on [Pro(30), Tyr(32), Leu(34)]NPY(28-36)-NH2 (BW1911U90). |
University Of Cincinnati And Va Medical Centers |
10866375 |
50 |
Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y5 receptor antagonists. |
Novartis Pharma |
9371234 |
49 |
Potent and selective 1,2,3-trisubstituted indole NPY Y-1 antagonists. |
Eli Lilly |