The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
28650658 |
54 |
Potent, Selective, and Cell Active Protein Arginine Methyltransferase 5 (PRMT5) Inhibitor Developed by Structure-Based Virtual Screening and Hit Optimization. |
Shandong University |
26220519 |
5 |
Design and synthesis of new non nucleoside inhibitors of DNMT3A. |
Unit£ |
25406944 |
20 |
Targeting DNA methylation with small molecules: what's next? |
Cnrs-Pierre Fabre |
25032507 |
43 |
Discovery of a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. |
University Of North Carolina At Chapel Hill |
24900829 |
11 |
Analogues of the Natural Product Sinefungin as Inhibitors of EHMT1 and EHMT2. |
University Of Copenhagen |
24387159 |
36 |
Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells. |
Sapienza University Of Rome |
23433670 |
15 |
Bromo-deaza-SAH: a potent and selective DOT1L inhibitor. |
Entremed |
23402879 |
1 |
Synthetic approaches to DNMT inhibitor SGI-1027 and effects on the U937 leukemia cell line. |
Universidade De Vigo |
24900432 |
51 |
Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2. |
TBA |
22854677 |
32 |
New cytosine derivatives as inhibitors of DNA methylation. |
Polish Academy Of Sciences |
22280363 |
104 |
Defining the mechanism of action and enzymatic selectivity of psammaplin A against its epigenetic targets. |
Imperial College |
22483584 |
3 |
Development of rationally designed DNA N6 adenine methyltransferase inhibitors. |
University Of Southampton |
21958292 |
7 |
Synthesis and biochemical evaluation ofd(2)-isoxazoline derivatives as DNA methyltransferase 1 inhibitors. |
Universit£ |
20006515 |
5 |
Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation. |
Deutsches Krebsforschungszentrum |
19364644 |
47 |
Constrained (l-)-S-adenosyl-l-homocysteine (SAH) analogues as DNA methyltransferase inhibitors. |
Methylgene |
19362833 |
41 |
SAR around (l)-S-adenosyl-l-homocysteine, an inhibitor of human DNA methyltransferase (DNMT) enzymes. |
Methylgene |
16420053 |
4 |
Discovery of two novel, small-molecule inhibitors of DNA methylation. |
Polish Academy Of Sciences |
28463515 |
21 |
Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells. |
Cnrs-Pierre Fabre Usr3388 |
27391855 |
24 |
Discovery of a Selective Covalent Inhibitor of Lysophospholipase-like 1 (LYPLAL1) as a Tool to Evaluate the Role of this Serine Hydrolase in Metabolism. |
Pfizer |