The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
27128184 |
13 |
Design, synthesis and biological evaluation of PSMA/hepsin-targeted heterobivalent ligands. |
Korea University |
27074627 |
4 |
Unprecedented Binding Mode of Hydroxamate-Based Inhibitors of Glutamate Carboxypeptidase II: Structural Characterization and Biological Activity. |
Academy Of Sciences Of The Czech Republic |
26894427 |
11 |
Preparation and Evaluation of Radiolabeled Antibody Recruiting Small Molecules That Target Prostate-Specific Membrane Antigen for Combined Radiotherapy and Immunotherapy. |
Mcmaster University |
25923815 |
11 |
Design of highly potent urea-based, exosite-binding inhibitors selective for glutamate carboxypeptidase II. |
Academy Of Sciences Of The Czech Republic |
22949627 |
3 |
Reversible disulfide formation of the glutamate carboxypeptidase II inhibitor E2072 results in prolonged systemic exposures in vivo. |
Johns Hopkins School Of Medicine |
25956413 |
12 |
Synthesis and evaluation of constrained phosphoramidate inhibitors of prostate-specific membrane antigen. |
Washington State University |
25822623 |
2 |
DUPA conjugation of a cytotoxic indenoisoquinoline topoisomerase I inhibitor for selective prostate cancer cell targeting. |
Purdue University |
24954515 |
21 |
Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. |
Academy Of Sciences Of The Czech Republic |
24354364 |
3 |
d-Thiolactones as prodrugs of thiol-based glutamate carboxypeptidase II (GCPII) inhibitors. |
Johns Hopkins University |
24063417 |
14 |
Preparation of asymmetric urea derivatives that target prostate-specific membrane antigen for SPECT imaging. |
Kyoto University |
23025786 |
28 |
Radiofluorinated derivatives of 2-(phosphonomethyl)pentanedioic acid as inhibitors of prostate specific membrane antigen (PSMA) for the imaging of prostate cancer. |
Bayer Healthcare |
22642259 |
22 |
Design, synthesis, and pharmacological evaluation of glutamate carboxypeptidase II (GCPII) inhibitors based on thioalkylbenzoic acid scaffolds. |
Eisai |
18023582 |
7 |
Phosphoramidate derivatives of hydroxysteroids as inhibitors of prostate-specific membrane antigen. |
Washington State University |
18060794 |
3 |
Design and synthesis of a siderophore conjugate as a potent PSMA inhibitor and potential diagnostic agent for prostate cancer. |
University Of Notre Dame |
21923190 |
10 |
Novel substrate-based inhibitors of human glutamate carboxypeptidase II with enhanced lipophilicity. |
Academy Of Sciences Of The Czech Republic |
22018464 |
4 |
Spacer length effects on in vitro imaging and surface accessibility of fluorescent inhibitors of prostate specific membrane antigen. |
Washington State University |
21074428 |
17 |
The discovery and structure-activity relationships of indole-based inhibitors of glutamate carboxypeptidase II. |
Eisai Research Institute |
20947349 |
3 |
A targeted low molecular weight near-infrared fluorescent probe for prostate cancer. |
Washington State University |
19897367 |
43 |
Bioisosterism of urea-based GCPII inhibitors: Synthesis and structure-activity relationship studies. |
Institutions |
| 8 |
Design and synthesis of novel monocyclic β-lactam inhibitors of prostate specific antigen |
TBA |
19111054 |
19 |
A series of halogenated heterodimeric inhibitors of prostate specific membrane antigen (PSMA) as radiolabeled probes for targeting prostate cancer. |
Molecular Insight Pharmaceuticals |
19108655 |
25 |
Multivalent scaffolds for affinity maturation of small molecule cell surface binders and their application to prostate tumor targeting. |
Justus-Liebig-Universitat Giessen |
19053825 |
6 |
Radiohalogenated prostate-specific membrane antigen (PSMA)-based ureas as imaging agents for prostate cancer. |
Institutions |
17869524 |
11 |
The molecular pruning of a phosphoramidate peptidomimetic inhibitor of prostate-specific membrane antigen. |
San Francisco State University |
12798312 |
22 |
Synthesis and biological evaluation of hydroxamate-Based inhibitors of glutamate carboxypeptidase II. |
Guilford Pharmaceuticals |
12723961 |
15 |
Synthesis and biological evaluation of thiol-based inhibitors of glutamate carboxypeptidase II: discovery of an orally active GCP II inhibitor. |
Guilford Pharmaceuticals |
11334560 |
18 |
Design, synthesis, and proposed active site binding analysis of monocyclic 2-azetidinone inhibitors of prostate specific antigen. |
University Of Oxford |
28759215 |
7 |
Discovery of a para-Acetoxy-benzyl Ester Prodrug of a Hydroxamate-Based Glutamate Carboxypeptidase II Inhibitor as Oral Therapy for Neuropathic Pain. |
Academy Of Sciences Of The Czech Republic |