The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
25794791 |
13 |
Recent advances in the chemistry and biology of pyridopyrimidines. |
Universit£ |
25259627 |
36 |
Structural basis for inhibition of mycobacterial and human adenosine kinase by 7-substituted 7-(Het)aryl-7-deazaadenine ribonucleosides. |
Academy Of Sciences Of The Czech Republic |
15149648 |
32 |
A TOPS-MODE approach to predict adenosine kinase inhibition. |
Vigo University |
18077363 |
314 |
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases. |
University Of Oxford |
15214773 |
76 |
Fragment-based drug discovery. |
Sunesis Pharmaceuticals |
8230132 |
7 |
New adenosine kinase inhibitors with oral antiinflammatory activity: synthesis and biological evaluation. |
University Of California |
3351857 |
1 |
Synthesis, intramolecular hydrogen bonding, and biochemical studies of clitocine, a naturally occurring exocyclic amino nucleoside. |
Nucleic Acid Research Institute |
21711054 |
16 |
Synthesis and significant cytostatic activity of 7-hetaryl-7-deazaadenosines. |
Academy Of Sciences Of The Czech Republic |
21319802 |
51 |
Non-nucleoside inhibitors of human adenosine kinase: synthesis, molecular modeling, and biological studies. |
Universita` Di Siena |
20055427 |
98 |
Fructose-1,6-bisphosphatase Inhibitors. 2. Design, synthesis, and structure-activity relationship of a series of phosphonic acid containing benzimidazoles that function as 5'-adenosinemonophosphate (AMP) mimics. |
Metabasis Therapeutics |
19348494 |
73 |
Fructose-1,6-bisphosphatase inhibitors. 1. Purine phosphonic acids as novel AMP mimics. |
Metabasis Therapeutics |
17197188 |
110 |
4-amino-5-aryl-6-arylethynylpyrimidines: structure-activity relationships of non-nucleoside adenosine kinase inhibitors. |
Abbott Laboratories |
16302820 |
45 |
Adenosine kinase inhibitors. 6. Synthesis, water solubility, and antinociceptive activity of 5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)pyrrolo[2,3-d]pyrimidines substituted at C4 with glycinamides and related compounds. |
Metabasis Therapeutics |
16190769 |
23 |
Adenosine kinase inhibitors. 5. Synthesis, enzyme inhibition, and analgesic activity of diaryl-erythro-furanosyltubercidin analogues. |
Metabasis Therapeutics |
15911258 |
45 |
Synthesis and biological evaluation of 6,7-disubstituted 4-aminopyrido[2,3-d]pyrimidines as adenosine kinase inhibitors. |
Abbott Laboratories |
15857145 |
22 |
Adenosine kinase inhibitors. 4. 6,8-Disubstituted purine nucleoside derivatives. Synthesis, conformation, and enzyme inhibition. |
Metabasis Therapeutics |
15261263 |
14 |
Synthesis and biological evaluation of pteridine and pyrazolopyrimidine based adenosine kinase inhibitors. |
Abbott Laboratories |
15050645 |
35 |
Discovery and optimization of 2-aryl oxazolo-pyrimidines as adenosine kinase inhibitors using liquid phase parallel synthesis. |
Bayer |
14613327 |
46 |
5,6,7-trisubstituted 4-aminopyrido[2,3-d]pyrimidines as novel inhibitors of adenosine kinase. |
Abbott Laboratories |
14561094 |
20 |
Adenosine kinase inhibitors. 3. Synthesis, SAR, and antiinflammatory activity of a series of l-lyxofuranosyl nucleosides. |
Metabasis Therapeutics |
12941329 |
30 |
Adenosine kinase inhibitors: polar 7-substitutent of pyridopyrimidine derivatives improving their locomotor selectivity. |
Abbott Laboratories |
11958989 |
32 |
QSAR study on adenosine kinase inhibition of pyrrolo[2,3-d]pyrimidine nucleoside analogues using the hansch approach. |
Jadavpur University |
11514141 |
16 |
Pyridopyrimidine analogues as novel adenosine kinase inhibitors. |
Abbott Laboratories |
11405650 |
42 |
Discovery of 4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin-3-yl)pyrido[2,3-d]pyrimidine, an orally active, non-nucleoside adenosine kinase inhibitor.. |
Abbott Laboratories |
11123986 |
5 |
Design of adenosine kinase inhibitors from the NMR-based screening of fragments. |
Abbott Laboratories |
10956197 |
34 |
Adenosine kinase inhibitors. 2. Synthesis, enzyme inhibition, and antiseizure activity of diaryltubercidin analogues. |
Metabasis Therapeutics |
10956196 |
39 |
Adenosine kinase inhibitors. 1. Synthesis, enzyme inhibition, and antiseizure activity of 5-iodotubercidin analogues. |
Metabasis Therapeutics |