The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
26741166 |
105 |
Discovery of (3-(4-(2-Oxa-6-azaspiro[3.3]heptan-6-ylmethyl)phenoxy)azetidin-1-yl)(5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-yl)methanone (AZD1979), a Melanin Concentrating Hormone Receptor 1 (MCHr1) Antagonist with Favorable Physicochemical Properties. |
Astrazeneca |
22542010 |
31 |
Discovery of a novel melanin concentrating hormone receptor 1 (MCHR1) antagonist with reduced hERG inhibition. |
Amgen |
19683441 |
33 |
Discovery of novel diarylketoxime derivatives as selective and orally active melanin-concentrating hormone 1 receptor antagonists. |
Tsukuba Research Institute |
22123324 |
36 |
Discovery and characterization of a potent and selective antagonist of melanin-concentrating hormone receptor 2. |
Amgen |
19500979 |
74 |
Optimization of 2-piperidin-4-yl-acetamides as melanin-concentrating hormone receptor 1 (MCH-R1) antagonists: Designing out hERG inhibition. |
Astrazeneca R & D M£Lndal |
19361985 |
17 |
Identification and characterization of a selective radioligand for melanin-concentrating hormone 1-receptor (MCH1R). |
Tsukuba Research Institute |
19403308 |
36 |
Discovery of novel spiro-piperidine derivatives as highly potent and selective melanin-concentrating hormone 1 receptor antagonists. |
Tsukuba Research Institute |
17448659 |
29 |
Design and synthesis of novel hydantoin-containing melanin-concentrating hormone receptor antagonists. |
Cerep |
17188866 |
17 |
Constrained 7-fluorocarboxychromone-4-aminopiperidine based Melanin-concentrating hormone receptor 1 antagonists: the effects of chirality on substituted indan-1-ylamines. |
Abbott Laboratories |
17178222 |
29 |
Quinazoline and benzimidazole MCH-1R antagonists. |
Argenta Discovery |
16919453 |
100 |
4-Aminoquinoline melanin-concentrating hormone 1-receptor (MCH1R) antagonists. |
Merck Research Laboratories |
16690312 |
110 |
Synthesis and structure-activity relationships of piperidine-based melanin-concentrating hormone receptor 1 antagonists. |
Schering-Plough Research Institute |
16202583 |
46 |
Biaryl diamides as potent melanin concentrating hormone receptor 1 antagonists. |
Schering-Plough Research Institute |
16134937 |
154 |
6-Acylamino-2-aminoquinolines as potent melanin-concentrating hormone 1 receptor antagonists. Identification, structure-activity relationship, and investigation of binding mode. |
7Tm Pharma |
15801820 |
31 |
Discovery of bicycloalkyl urea melanin concentrating hormone receptor antagonists: orally efficacious antiobesity therapeutics. |
Schering-Plough Research Institute |
15380202 |
85 |
4-Acylamino-and 4-ureidobenzamides as melanin-concentrating hormone (MCH) receptor 1 antagonists. |
7Tm Pharma |
26915401 |
1 |
A Novel Inhibitor of the Obesity-Related Protein FTO. |
Basic Medical College Of Zhengzhou University |