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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28650658 54 Potent, Selective, and Cell Active Protein Arginine Methyltransferase 5 (PRMT5) Inhibitor Developed by Structure-Based Virtual Screening and Hit Optimization.EBI Shandong University
26220519 5 Design and synthesis of new non nucleoside inhibitors of DNMT3A.EBI Unit£ de Service et de Recherche CNRS-Pierre Fabre n£3388
25406944 20 Targeting DNA methylation with small molecules: what's next?EBI CNRS-Pierre Fabre
25032507 43 Discovery of a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.EBI University of North Carolina at Chapel Hill
24900829 11 Analogues of the Natural Product Sinefungin as Inhibitors of EHMT1 and EHMT2.EBI University of Copenhagen
24387159 36 Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells.EBI Sapienza Universit£ di Roma
23433670 15 Bromo-deaza-SAH: a potent and selective DOT1L inhibitor.EBI EntreMed Inc.
23402879 1 Synthetic approaches to DNMT inhibitor SGI-1027 and effects on the U937 leukemia cell line.EBI Universidade de Vigo
24900432 51 Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2.EBI TBA
22854677 32 New cytosine derivatives as inhibitors of DNA methylation.EBI Polish Academy of Sciences
22280363 104 Defining the mechanism of action and enzymatic selectivity of psammaplin A against its epigenetic targets.EBI Imperial College London
22483584 3 Development of rationally designed DNA N6 adenine methyltransferase inhibitors.EBI University of Southampton
21958292 7 Synthesis and biochemical evaluation ofd(2)-isoxazoline derivatives as DNA methyltransferase 1 inhibitors.EBI Universit£ degli Studi di Salerno
20006515 5 Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation.EBI Deutsches Krebsforschungszentrum
19364644 47 Constrained (l-)-S-adenosyl-l-homocysteine (SAH) analogues as DNA methyltransferase inhibitors.EBI MethylGene Inc.
19362833 41 SAR around (l)-S-adenosyl-l-homocysteine, an inhibitor of human DNA methyltransferase (DNMT) enzymes.EBI MethylGene Inc.
16420053 4 Discovery of two novel, small-molecule inhibitors of DNA methylation.EBI Polish Academy of Sciences
28463515 21 Rational Design of Bisubstrate-Type Analogues as Inhibitors of DNA Methyltransferases in Cancer Cells.EBI CNRS-Pierre Fabre USR3388
27391855 24 Discovery of a Selective Covalent Inhibitor of Lysophospholipase-like 1 (LYPLAL1) as a Tool to Evaluate the Role of this Serine Hydrolase in Metabolism.BDB Pfizer Inc.