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34 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
2785211 18 Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist.EBI Johns Hopkins Medical Institutions
3020246 11 Irreversible blockage of opioid receptor types by ester homologues of beta-funaltrexamine.EBI TBA
3020245 4 Synthesis and biological activity of analogues of beta-chlornaltrexamine and beta-funaltrexamine at opioid receptors.EBI TBA
6319699 5 Replacement of the peptide-backbone amides connecting Tyr-Gly and Gly-Gly in leucine-enkephalin with ketomethylene groups: synthesis and biological activity.EBI TBA
6209395 8 Diastereomeric 6-desoxy-6-spiro-alpha-methylene-gamma-butyrolactone derivatives of naltrexone and oxymorphone. Selective irreversible inhibition of naltrexone binding in an opioid receptor preparation by a conformationally restricted michael acceptor ligand.EBI TBA
6292421 6 N-Methylnalorphine: definition of N-allyl conformation for antagonism at the opiate receptor.EBI TBA
6292420 6 Synthesis and pharmacology of metabolically stable tert-butyl ethers of morphine and levorphanol.EBI TBA
26346669 53 Synthesis of new opioid derivatives with a propellane skeleton and their pharmacologies: Part 5, novel pentacyclic propellane derivatives with a 6-amide side chain.EBI University of Tsukuba
26252963 15 Novel diazabicycloalkane delta opioid agonists.EBI Istituto di Farmacologia Traslazionale
25783191 87 Design, syntheses, and pharmacological characterization of 17-cyclopropylmethyl-3,14-dihydroxy-4,5a-epoxy-6a-(isoquinoline-3'-carboxamido)morphinan analogues as opioid receptor ligands.EBI Virginia Commonwealth University
23116891 15 Synthesis of new opioid derivatives with a propellane skeleton and their pharmacologies: part 3, novel propellane derivatives with pentacyclic skeletons.EBI Kitasato University
22734622 78 Synthesis and evaluation of aryl-naloxamide opiate analgesics targeting truncated exon 11-associatedµ opioid receptor (MOR-1) splice variants.EBI Memorial Sloan-Kettering Cancer Center
18829333 28 Design, synthesis, and structure-activity relationship of novel opioid kappa-agonists.EBI Toray Industries, Inc.
17702750 1 Long-acting kappa opioid antagonists disrupt receptor signaling and produce noncompetitive effects by activating c-Jun N-terminal kinase.EBI University of Washington
10891118 6 Enkephalin glycopeptide analogues produce analgesia with reduced dependence liability.EBI University of Northern Colorado
9379438 31 Discovery of a novel class of substituted pyrrolooctahydroisoquinolines as potent and selective delta opioid agonists, based on an extension of the message-address concept.EBI SmithKline Beecham S.p.A.
9207938 15 Pyrrolomorphinans as delta opioid receptor antagonists. The role of steric hindrance in conferring selectivity.EBI University of Minnesota
9171881 17 7-Spiroindanyl derivatives of naltrexone and oxymorphone as selective ligands for delta opioid receptors.EBI University of Minnesota
8648612 30 Arylacetamide-derived fluorescent probes: synthesis, biological evaluation, and direct fluorescent labeling of kappa opioid receptors in mouse microglial cells.EBI University of Minnesota
1333013 29 Opioid agonist and antagonist activities of morphindoles related to naltrindole.EBI University of Minnesota
2549247 39 Benzofuro[2,3-c]pyridin-6-ols: synthesis, affinity for opioid-receptor subtypes, and antinociceptive activity.EBI CIBA-GEIGY Corporation
 36 Pyrrolooctahydroisoquinolines as potent and selective opioid receptor ligands: SAR analysis and docking studiesEBI TBA
21392859 1 Synthesis and biological evaluation of dibenz[b,f][1,5]oxazocine derivatives for agonist activity at κ-opioid receptor.EBI Indian Institute of Chemical Biology
 26 6N-Cinnamoyl-β-naltrexamine and its p-nitro derivative. High efficacy κ-opioid agonists with weak antagonist actionsEBI TBA
12408719 21 Synthesis and structure-activity relationships of an orally available and long-acting analgesic peptide, N(alpha)-amidino-Tyr-D-Arg-Phe-MebetaAla-OH (ADAMB).EBI Daiichi Fine Chemical Co. Ltd.
11150174 84 Synthesis and in vitro and in vivo activity of (-)-(1R,5R,9R)- and (+)-(1S,5S,9S)-N-alkenyl-, -N-alkynyl-, and -N-cyanoalkyl-5, 9-dimethyl-2'-hydroxy-6,7-benzomorphan homologues.EBI Virginia Commonwealth University
9301669 24 7-spirobenzocyclohexyl derivatives of naltrexone, oxymorphone, and hydromorphone as selective opioid receptor ligands.EBI University of Minnesota
8410989 58 Structure-affinity relationship studies on 5-HT1A receptor ligands. 1. Heterobicyclic phenylpiperazines with N4-alkyl substituents.EBI Solvay Duphar Research Laboratories
7932577 24 Selective kappa-opioid agonists: synthesis and structure-activity relationships of piperidines incorporating on oxo-containing acyl group.EBI SmithKline Beecham Farmaceutici S.p.A.
1972964 40 Design and synthesis of highly potent and selective cyclic dynorphin A analogues.EBI University of Arizona
1967312 91 Synthesis and structure-activity relationships of dynorphin A-(1-8) amide analogues.EBI Eisai Co., Ltd.
1648141 21 Naphtho and benzo analogues of the kappa opioid agonist trans-(+/-)-3,4-dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl] benzeneacetamide.EBI University of Notre Dame
26520885 21 Synthesis of 4-thiazolidinone analogs as potent in vitro anti-urease agents.BDB Hazara University