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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27690432 75 Discovery of Second Generation Reversible Covalent DPP1 Inhibitors Leading to an Oxazepane Amidoacetonitrile Based Clinical Candidate (AZD7986).EBI CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
24913985 73 SAR studies of differently functionalized chalcones based hydrazones and their cyclized derivatives as inhibitors of mammalian cathepsin B and cathepsin H.EBI Kurukshetra University
24642566 17 Acyl hydrazides and triazoles as novel inhibitors of mammalian cathepsin B and cathepsin H.EBI Kurukshetra University
23252745 86 Development of new cathepsin B inhibitors: combining bioisosteric replacements and structure-based design to explore the structure-activity relationships of nitroxoline derivatives.EBI University of Ljubljana
19715320 87 Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI University of Florida
19419206 77 Identification of 3-acetyl-2-aminoquinolin-4-one as a novel, nonpeptidic scaffold for specific calpain inhibitory activity.EBI Ewha Womans University
17535802 91 Inhibition of the activation of multiple serine proteases with a cathepsin C inhibitor requires sustained exposure to prevent pro-enzyme processing.EBI Merck Research Laboratories
18226527 80 The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K.EBI Merck Frosst Centre for Therapeutic Research
19665376 48 Design and synthesis of dipeptidyl nitriles as potent, selective, and reversible inhibitors of cathepsin C.EBI Merck Frosst Canada& Co.
18313933 18 Substrate optimization for monitoring cathepsin C activity in live cells.EBI Genomics Institute of the Novartis Research Foundation (GNF)
17196818 90 Bicyclic carbamates as inhibitors of papain-like cathepsin proteases.EBI The Genomics Institute of the Novartis Research Foundation
16647256 16 Dipeptidyl nitriles as human dipeptidyl peptidase I inhibitors.EBI Arpida A/S
16290936 69 Semicarbazone-based inhibitors of cathepsin K, are they prodrugs for aldehyde inhibitors?EBI GlaxoSmithKline
15896958 32 Acyclic cyanamide-based inhibitors of cathepsin K.EBI GlaxoSmithKline
15837295 55 A structural screening approach to ketoamide-based inhibitors of cathepsin K.EBI GlaxoSmithKline
15780613 28 Novel and potent cyclic cyanamide-based cathepsin K inhibitors.EBI GlaxoSmithKline
15341947 57 Potent and selective P2-P3 ketoamide inhibitors of cathepsin K with good pharmacokinetic properties via favorable P1', P1, and/or P3 substitutions.EBI GlaxoSmithKline
10052963 7 New peptidic cysteine protease inhibitors derived from the electrophilic alpha-amino acid aziridine-2,3-dicarboxylic acid.EBI Albert-Ludwigs-University of Freiburg