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46 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
24915003 34 Probing of primed and unprimed sites of calpains: Design, synthesis and evaluation of epoxysuccinyl-peptide derivatives as selective inhibitors.EBI E£tv£s Lor£nd University (ELTE)
23834438 10 Design, synthesis, and optimization of novel epoxide incorporating peptidomimetics as selective calpain inhibitors.EBI University of Illinois College of Pharmacy
1597856 20 Ester and amide derivatives of E64c as inhibitors of platelet calpains.EBI State University of New York Health Science Center
19715320 87 Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation.EBI University of Florida
18396356 13 Design and synthesis of calpain inhibitory 6-pyridone 2-carboxamide derivatives.EBI Kyung Hee University
19419206 77 Identification of 3-acetyl-2-aminoquinolin-4-one as a novel, nonpeptidic scaffold for specific calpain inhibitory activity.EBI Ewha Womans University
19041242 25 Design and synthesis of 4-aryl-4-oxobutanoic acid amides as calpain inhibitors.EBI Shenyang Pharmaceutical University
10669559 180 Protease inhibitors: current status and future prospects.EBI University of Queensland
9667954 47 D-amino acid containing, high-affinity inhibitors of recombinant human calpain I.EBI Cephalon, Inc.
14980679 30 Dipeptidyl aspartyl fluoromethylketones as potent caspase-3 inhibitors: SAR of the P2 amino acid.EBI Maxim Pharmaceuticals
15013018 47 1,2-Benzothiazine 1,1-dioxide alpha-ketoamide analogues as potent calpain I inhibitors.EBI Cephalon, Inc.
10476870 9 Hydroxyoxazolidines as alpha-aminoacetaldehye equivalents: novel inhibitors of calpain.EBI Hoechst Marion Roussel, Inc.
21504847 12 Synthesis of cinnamoyl ketoamides as hybrid structures of antioxidants and calpain inhibitors.EBI College of Pharmacy Kyung Hee University
20690647 33 Peptidyl alpha-ketoamides with nucleobases, methylpiperazine, and dimethylaminoalkyl substituents as calpain inhibitors.EBI Georgia Institute of Technology
 65 Subsite requirements for peptide aldehyde inhibitors of human calpain IEBI TBA
 10 Nonpeptidic inhibitors of recombinant human calpain IEBI TBA
 2 Oligopresentation of protease inhibitors with β-cyclodextrin as templateEBI TBA
 6 Xanthene derived potent nonpeptidic inhibitors of recombinant human calpain IEBI TBA
 1 Synthesis of cystamidin a (pyrrole-3-propanamide), a reported calpain inhibitorEBI TBA
 22 Inhibition of human erythrocyte calpain I by novel quinolinecarboxamidesEBI TBA
18789863 10 Molecular design to enhance the penetration into the retina via ocular instillation.EBI Senju Pharmaceutical Co., Ltd
18694642 6 Synthesis and calpain inhibitory activity of peptidomimetic compounds with constrained amino acids at the P2 position.EBI The University of Tennessee Health Science Center
18024028 14 Design and synthesis of 4-quinolinone 2-carboxamides as calpain inhibitors.EBI Kyung Hee University
16913717 42 Synthesis, calpain inhibitory activity, and cytotoxicity of P2-substituted proline and thiaproline peptidyl aldehydes and peptidyl alpha-ketoamides.EBI The University of Tennessee Health Science Center
16789748 31 Exploration of orally available calpain inhibitors 2: peptidyl hemiacetal derivatives.EBI Senju Pharmaceutical Company, Ltd.
15911268 13 Synthesis and biological evaluation of chromone carboxamides as calpain inhibitors.EBI Institute of Science & Technology
15713391 19 Dipeptidyl aspartyl fluoromethylketones as potent caspase inhibitors: peptidomimetic replacement of the P2 alpha-amino acid by a alpha-hydroxy acid.EBI Maxim Pharmaceuticals
15634028 5 Retro hydrazino-azapeptoids as peptidomimetics of proteasome inhibitors.EBI Université Rennes 1
15203170 7 Novel dual inhibitors of calpain and lipid peroxidation.EBI Institut Henri Beaufour
12773044 18 Benzoylalanine-derived ketoamides carrying vinylbenzyl amino residues: discovery of potent water-soluble calpain inhibitors with oral bioavailability.EBI Abbott GmbH & Co. KG
12593666 30 Structure-activity relationship study and drug profile of N-(4-fluorophenylsulfonyl)-L-valyl-L-leucinal (SJA6017) as a potent calpain inhibitor.EBI Senju Pharmaceutical Co.
12039572 7 Exploration of peptidyl hydrazones as water-soluble calpain inhibitors.EBI Senju Pharmaceutical Co., Ltd.
11992771 19 Discovery of phenyl alanine derived ketoamides carrying benzoyl residues as novel calpain inhibitors.EBI Abbott GmbH&Co. KG
11585453 52 1,2-Benzothiazine 1,1-dioxide P(2)-P(3) peptide mimetic aldehyde calpain I inhibitors.EBI Cephalon, Inc.
11551769 2 Synthesis of a reported calpain inhibitor isolated from Streptomyces griseus.EBI The University of Tennessee Health Science Center
11551762 16 Potent peptide alpha-ketohydroxamate inhibitors of recombinant human calpain I.EBI Cephalon, Inc.
11012026 18 Synthesis and biological evaluation of novel piperidine carboxamide derived calpain inhibitors.EBI KNOLL AG
10476871 22 P2-achiral, P'-extended alpha-ketoamide inhibitors of calpain I.EBI Cephalon Inc.
10021915 3 The synthesis of ketomethylene pseudopeptide analogues of dipeptide aldehyde inhibitors of calpain.EBI Hoechst Marion Roussel, Inc.
9873596 18 P2-proline-derived inhibitors of calpain I.EBI Cephalon, Inc.
9748367 11 Novel peptidyl phosphorus derivatives as inhibitors of human calpain I.EBI Cephalon, Inc.
8831774 261 Novel peptidyl alpha-keto amide inhibitors of calpains and other cysteine proteases.EBI School of Chemistry and Biochemistry
8071940 32 Stereospecific synthesis of peptidyl alpha-keto amides as inhibitors of calpain.EBI Alkermes, Inc.
24095934 60 Synthesis and investigation of dihydroxychalcones as calpain and cathepsin inhibitors.BDB Ewha Womans University, Seoul 120-750, Republic of Korea.
18636690 11 Structural basis for the potent calpain inhibitory activity of peptidyl alpha-ketoacids.BDB University of Tennessee Health Science Center