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62 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
592327 104 Potent reversible anticholinesterase agents. Bis- and mono-N-substituted benzoquinolinium halides.EBI TBA
23151013 56 Carbamate derivatives of indolines as cholinesterase inhibitors and antioxidants for the treatment of Alzheimer's disease.EBI Bar Ilan University
22503231 66 Multipotent MAO and cholinesterase inhibitors for the treatment of Alzheimer's disease: synthesis, pharmacological analysis and molecular modeling of heterocyclic substituted alkyl and cycloalkyl propargyl amine.EBI Laboratorio de Radicales Libres y Qu�mica Computacional (IQOG, CSIC)
22445674 43 Cholinestrase inhibitory effects of geranylated flavonoids from Paulownia tomentosa fruits.EBI Graduate School of Gyeongsang National University
18406135 22 Design and synthesis of tacrine-ferulic acid hybrids as multi-potent anti-Alzheimer drug candidates.EBI Friedrich-Schiller-Universit£t Jena
17854153 2 Brunneins A-C, beta-carboline alkaloids from Cortinarius brunneus.EBI Institute of Plant Biochemistry
17451950 36 Derivatives of oxoisoaporphine alkaloids: a novel class of selective acetylcholinesterase inhibitors.EBI Sun Yat-Sen University
15633997 18 Propidium-based polyamine ligands as potent inhibitors of acetylcholinesterase and acetylcholinesterase-induced amyloid-beta aggregation.EBI University of Bologna
11831902 12 Pyridophens: binary pyridostigmine-aprophen prodrugs with differential inhibition of acetylcholinesterase, butyrylcholinesterase, and muscarinic receptors.EBI Institute of Research
9873615 9 Conformationally restricted carbamate inhibitors of horse serum butyrylcholinesterase.EBI National Chung-Hsing University
22041172 41 Benzenediol-berberine hybrids: multifunctional agents for Alzheimer's disease.EBI Guangzhou Institute of Biomedicine and Health
21975066 59 Formulating a new basis for the treatment against botulinum neurotoxin intoxication: 3,4-Diaminopyridine prodrug design and characterization.EBI The Scripps Research Institute
21417225 116 Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity.EBI Universidad de Granada
21429752 72 Design, synthesis and structure-activity relationship (SAR) studies of 2,4-disubstituted pyrimidine derivatives: dual activity as cholinesterase and A β-aggregation inhibitors.EBI University of Waterloo
21397508 36 Synthesis, biological evaluation and molecular modeling of novel triazole-containing berberine derivatives as acetylcholinesterase and β-amyloid aggregation inhibitors.EBI Sun Yat-sen University
21211982 30 Design, synthesis and evaluation of novel tacrine-multialkoxybenzene hybrids as dual inhibitors for cholinesterases and amyloid beta aggregation.EBI Sun Yat-sen University
20880702 35 Berberine derivatives, with substituted amino groups linked at the 9-position, as inhibitors of acetylcholinesterase/butyrylcholinesterase.EBI Sun Yat-sen University
20656495 56 Multipotent drugs with cholinergic and neuroprotective properties for the treatment of Alzheimer and neuronal vascular diseases. I. Synthesis, biological assessment, and molecular modeling of simple and readily available 2-aminopyridine-, and 2-chloropyridine-3,5-dicarbonitriles.EBI Laboratorio de Radicales Libres y Química Computacional (IQOG, CSIC)
 39 The synthesis and in vitro acetylcholinesterase and butyrylcholinesterase inhibitory activity of tacrine (Cognex®) derivatiesEBI TBA
19053746 22 NO-donating tacrine hybrid compounds improve scopolamine-induced cognition impairment and show less hepatotoxicity.EBI Friedrich Schiller University Jena
18343673 39 Design, synthesis and pharmacological evaluation of hybrid molecules out of quinazolinimines and lipoic acid lead to highly potent and selective butyrylcholinesterase inhibitors with antioxidant properties.EBI Friedrich-Schiller-Universität Jena
17317172 9 Methyl 2-(2-(4-formylphenoxy)acetamido)-2-substituted acetate derivatives: a new class of acetylcholinesterase inhibitors.EBI Sun Yat-sen University
16942014 32 Homobivalent quinazolinimines as novel nanomolar inhibitors of cholinesterases with dirigible selectivity toward butyrylcholinesterase.EBI Friedrich-Schiller-Universität Jena
16274989 40 Isolation and cholinesterase-inhibition studies of sterols from Haloxylon recurvum.EBI University of Karachi
14611850 8 Cage amines as the stopper inhibitors of cholinesterases.EBI National Chung-Hsing University
8064800 32 Novel benzisoxazole derivatives as potent and selective inhibitors of acetylcholinesterase.EBI Pfizer Inc.
22871134 34 Design, synthesis and evaluation of new thiazole-piperazines as acetylcholinesterase inhibitors.BDB Anadolu University
22630076 38 Synthesis and anticholinesterase activities of novel 1,3,4-thiadiazole based compounds.BDB University of Life Sciences
22380775 28 2-(2-indolyl-)-4(3H)-quinazolines derivates as new inhibitors of AChE: design, synthesis, biological evaluation and molecular modelling.BDB Sun Yat-sen University
20233015 6 Nostotrebin 6, a bis(cyclopentenedione) with cholinesterase inhibitory activity isolated from Nostoc sp. str. Lukesová 27/97.BDB Brno University of Technology
20030505 6 Stereoselective inhibition of butyrylcholinesterase by enantiomers of exo- and endo-2-norbornyl-N-n-butylcarbamates.BDB Chung Shan Medical University Hospital
28501648 14 Tetrahydroacridine derivatives with fluorobenzoic acid moiety as multifunctional agents for Alzheimer's disease treatment.BDB Medical University of Lodz
 18 Efficient synthesis of novel dialkyl-3-cyanopropylphosphate derivatives and evaluation of their anticholinesterase activityBDB University of Carthage
 68 Synthesis, crystal structure determination, biological screening and docking studies of N1-substituted derivatives of 2,3-dihydroquinazolin-4(1H)-one as inhibitors of cholinesterases.BDB University of Sargodha
 18 Novel multi-targeted agents for Alzheimer's disease: Synthesis, biological evaluation, and molecular modeling of novel 2-[4-(4-substitutedpiperazin-1-yl)phenyl]benzimidazolesBDB Hacettepe University
27863021 30 Synthesis and anticholinesterase activity of new substituted benzo[d]oxazole-based derivatives.BDB Shahid Bahonar University of Kerman
28245905 70 Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity.BDB Charles University
28126287 50 Synthesis, biological evaluation and docking studies of 2,3-dihydroquinazolin-4(1H)-one derivatives as inhibitors of cholinesterases.BDB University of Sargodha
27914694 32 Synthesis of novel chromenones linked to 1,2,3-triazole ring system: Investigation of biological activities against Alzheimer's disease.BDB Tehran University of Medical Sciences
27434226 140 Evaluation of multifunctional synthetic tetralone derivatives for treatment of Alzheimer's disease.BDB Wuhan University of Technology
27085663 30 Novel N-allyl/propargyl tetrahydroquinolines: Synthesis via Three-component Cationic Imino Diels-Alder Reaction, Binding Prediction, and Evaluation as Cholinesterase Inhibitors.BDB Universidad de Talcaa
27750058 46 Rational design and synthesis of dihydropyrimidine based dual binding site acetylcholinesterase inhibitors.BDB Hazara University
27289559 38 Design and synthesis of novel anti-Alzheimer's agents: Acridine-chromenone and quinoline-chromenone hybrids.BDB Tehran University of Medical Sciences
27231829 34 New cholinesterase inhibitors for Alzheimer's disease: Structure Activity Studies (SARs) and molecular docking of isoquinolone and azepanone derivatives.BDB Universidade de Évora
26851737 36 One-pot synthesis of tetrazole-1,2,5,6-tetrahydronicotinonitriles and cholinesterase inhibition: Probing the plausible reaction mechanism via computational studies.BDB University of Karachi
26440714 28 Synthesis, cholinesterase inhibition and molecular modelling studies of coumarin linked thiourea derivatives.BDB Quaid-I-Azam University
26077890 33 Design, Synthesis, Biological Evaluation, and Docking Study of Acetylcholinesterase Inhibitors: New Acridone-1,2,4-oxadiazole-1,2,3-triazole Hybrids.BDB Tehran University of Medical Sciences
26010139 34 Synthesis and anticholinergic activity of 4-hydroxycoumarin derivatives containing substituted benzyl-1,2,3-triazole moiety.BDB Tehran University of Medical Sciences
25951978 38 Syntheses, cholinesterases inhibition, and molecular docking studies of pyrido[2,3-b]pyrazine derivatives.BDB University of Karachi
26042530 40 Discovery of isoalloxazine derivatives as a new class of potential anti-Alzheimer agents and their synthesis.BDB The M. S. University of Baroda
25706320 86 Synthesis, antioxidant and anticholinesterase activities of novel coumarylthiazole derivatives.BDB Bezmialem Vakif University
25462625 58 Salicylanilide diethyl phosphates as cholinesterases inhibitors.BDB Charles University in Prague
21621811 10 Synthesis and biological activity of derivatives of tetrahydroacridine as acetylcholinesterase inhibitors.BDB Medical University of Lodz
18569333 14 Butyrylcholinesterase, lipoxygenase inhibiting and antifungal alkaloids from Isatis tinctoria.BDB PCSIR Laboratories Complex
17252943 10 New natural cholinesterase inhibiting and calcium channel blocking quinoline alkaloids.BDB University of Karachi
15895683 14 Synthesis and inhibitory potential towards acetylcholinesterase, butyrylcholinesterase and lipoxygenase of some variably substituted chalcones.BDB Quaid-i-Azam University
16530804 4 3-Amidoquinuclidine derivatives: synthesis of compounds and inhibition of butyrylcholinesterase.BDB University of Zagreb
12431053 293 Novel dual inhibitors of AChE and MAO derived from hydroxy aminoindan and phenethylamine as potential treatment for Alzheimer's disease.BDB Teva Pharmaceutical Industries
11425559 24 Novel and potent tacrine-related hetero- and homobivalent ligands for acetylcholinesterase and butyrylcholinesterase.BDB Universita degli Studi di Siena
16420031 46 Novel tacrine-melatonin hybrids as dual-acting drugs for Alzheimer disease, with improved acetylcholinesterase inhibitory and antioxidant properties.BDB Instituto de Quimica Medica (CSIC)
15771436 38 Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors.BDB Universita di Siena