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19 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27994766 28 Discovery of New Bromodomain Scaffolds by Biosensor Fragment Screening.EBI University of Dundee
27682507 167 Discovery of a Potent and Selective in Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300.EBI Genentech
26701186 50 KATching-Up on Small Molecule Modulators of Lysine Acetyltransferases.EBI University of Freiburg
26731131 2 Structure-Based Identification of Inhibitory Fragments Targeting the p300/CBP-Associated Factor Bromodomain.EBI University of Oxford
26230603 176 Structure-Based Optimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors.EBI GlaxoSmithKline
25730130 20 A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach.EBI Universit£ degli Studi di Salerno
25249180 146 The discovery of I-BET726 (GSK1324726A), a potent tetrahydroquinoline ApoA1 up-regulator and selective BET bromodomain inhibitor.EBI GlaxoSmithKline R&D
24345448 4 Azide-alkyne cycloaddition affording enzymatically tunable bisubstrate based inhibitors of histone acetyltransferase PCAF.EBI Utrecht University
24144283 100 Structure-guided design of potent diazobenzene inhibitors for the BET bromodomains.EBI Icahn School of Medicine at Mount Sinai
22924434 4 Progress in the development and application of small molecule inhibitors of bromodomain-acetyl-lysine interactions.EBI University of Oxford
19114310 30 Bisubstrate Inhibitors of the MYST HATs Esa1 and Tip60.EBI Georgia State University
19101154 28 Synthesis of isothiazol-3-one derivatives as inhibitors of histone acetyltransferases (HATs).EBI Institute of Cancer Research
22100137 6 6-alkylsalicylates are selective Tip60 inhibitors and target the acetyl-CoA binding site.EBI University of Groningen
21353783 37 Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitors.EBI Albert-Ludwigs-University of Freiburg
20655754 2 Improved inhibition of the histone acetyltransferase PCAF by an anacardic acid derivative.EBI Groningen Research Institute of Pharmacy
19683843 16 Reactivity of isothiazolones and isothiazolone-1-oxides in the inhibition of the PCAF histone acetyltransferase.EBI University of Groningen
19111471 19 Inhibition of the PCAF histone acetyl transferase and cell proliferation by isothiazolones.EBI University of Groningen