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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27448773 16 Steric structure-activity relationship of cyproheptadine derivatives as inhibitors of histone methyltransferase Set7/9.EBI Tokyo Medical and Dental University (TMDU)
27088648 5 Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription.EBI RIKEN
26390175 10 Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening.EBI Shanghai University
25406853 72 Selective inhibitors of protein methyltransferases.EBI Icahn School of Medicine at Mount Sinai
25746813 37 SAH derived potent and selective EZH2 inhibitors.EBI Pfizer Inc.
25032507 43 Discovery of a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.EBI University of North Carolina at Chapel Hill
25333769 22 Identifying novel selective non-nucleoside DNA methyltransferase 1 inhibitors through docking-based virtual screening.EBI Chinese Academy of Sciences
24650704 6 Using 'biased-privileged' scaffolds to identify lysine methyltransferase inhibitors.EBI Rockefeller University
20219369 5 Toward the development of potent and selective bisubstrate inhibitors of protein arginine methyltransferases.EBI University Park
21780790 65 Optimization of cellular activity of G9a inhibitors 7-aminoalkoxy-quinazolines.EBI University of North Carolina at Chapel Hill
21612300 30 Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity.EBI The University of Texas MD Anderson Cancer Center
21440447 15 Acyl derivatives of p-aminosulfonamides and dapsone as new inhibitors of the arginine methyltransferase hPRMT1.EBI Albert-Ludwigs-University of Freiburg
20614940 76 Protein lysine methyltransferase G9a inhibitors: design, synthesis, and structure activity relationships of 2,4-diamino-7-aminoalkoxy-quinazolines.EBI University of North Carolina at Chapel Hill
19836951 33 1,2-Diamines as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1).EBI MethylGene Inc
28135235 71 An allosteric PRC2 inhibitor targeting the H3K27me3 binding pocket of EED.BDB Novartis Institutes for BioMedical Research