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13 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27589480 72 Design and Synthesis of an Investigational Nonapeptide KISS1 Receptor (KISS1R) Agonist, Ac-d-Tyr-Hydroxyproline (Hyp)-Asn-Thr-Phe-azaGly-Leu-Arg(Me)-Trp-NHEBI Takeda Pharmaceutical Company Ltd
25811530 20 Rational design of triazololipopeptides analogs of kisspeptin inducing a long-lasting increase of gonadotropins.EBI UMR7247; Universit£ Fran£ois Rabelais Tours; IFCE)
24918545 81 Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.EBI Takeda Pharmaceutical Company Ltd.
24047141 64 Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity.EBI Takeda Pharmaceutical Company Ltd
22995619 22 Trypsin resistance of a decapeptide KISS1R agonist containing an N¿-methylarginine substitution.EBI Takeda Pharmaceutical Company Ltd
22975302 45 Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.EBI Takeda Pharmaceutical Company Ltd
20580563 42 2-acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats.EBI Takeda Pharmaceutical Company, Ltd
20457527 42 Synthesis and structure-activity relationships of 2-acylamino-4,6-diphenylpyridine derivatives as novel antagonists of GPR54.EBI Takeda Pharmaceutical Company, Ltd
17579384 27 SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54.EBI Kyoto University
17266198 84 Metastin (KiSS-1) mimetics identified from peptide structure-activity relationship-derived pharmacophores and directed small molecule database screening.EBI University of Minnesota Health Science Center
19007202 12 Development of Novel G-Protein-Coupled Receptor 54 Agonists with Resistance to Degradation by Matrix Metalloproteinase.BDB Kyoto University