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12 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27682507 167 Discovery of a Potent and Selective in Vivo Probe (GNE-272) for the Bromodomains of CBP/EP300.EBI Genentech
27326325 44 GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain.EBI GlaxoSmithKline
27167503 17 Twenty Crystal Structures of Bromodomain and PHD Finger Containing Protein 1 (BRPF1)/Ligand Complexes Reveal Conserved Binding Motifs and Rare Interactions.EBI University of Z£rich
26982797 20 The"Gatekeeper" Residue Influences the Mode of Binding of Acetyl Indoles to Bromodomains.EBI University of Z£rich
26731611 30 4-Acyl Pyrrole Derivatives Yield Novel Vectors for Designing Inhibitors of the Acetyl-Lysine Recognition Site of BRD4(1).EBI Albert-Ludwigs-Universit£t Freiburg
26572217 60 Disrupting Acetyl-Lysine Recognition: Progress in the Development of Bromodomain Inhibitors.EBI Genentech
26061247 71 Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor.EBI The University of Texas MD Anderson Cancer Center
25974391 78 Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF.EBI University of Oxford
26230603 176 Structure-Based Optimization of Naphthyridones into Potent ATAD2 Bromodomain Inhibitors.EBI GlaxoSmithKline
25408830 43 1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain.EBI GlaxoSmithKline
25249180 146 The discovery of I-BET726 (GSK1324726A), a potent tetrahydroquinoline ApoA1 up-regulator and selective BET bromodomain inhibitor.EBI GlaxoSmithKline R&D
28849908 13 Selective Targeting of Bromodomains of the Bromodomain-PHD Fingers Family Impairs Osteoclast Differentiation.BDB Oxford University