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Compounds Sorted by Binding Targets per Compound

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190   253   269   272   278   297   310   314   332   362   363   364   365   366   367   368   370   371   372   374   375   
376   378   379   380   383   384   385   386   388   389   391   393   394   397   406   411   412   413   415   427   434   
Compounds Sorted Alphabetically
Compound Name
(alphabetical)
Binding TargetsEnz. Inhib. DataITC DataAlternate Compound Names
KiIC50KdEC50KoffKonOther
BDBM86201
PNG
  • 5-Hydroxytryptamine receptor 6 (5-HT6)
  • 5-Hydroxytryptamine receptor 7 (5-HT7)
  • 5-hydroxytryptamine receptor 1A (5-HT1A)
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 3A
  • ADRB2
  • Adrenergic alpha1B
  • Adrenergic receptor beta
  • Alpha-1A adrenergic receptor
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • Alpha-2C adrenergic receptor
  • CHRM5
  • Calcium channel
  • Cannabinoid receptor 1
  • Cholinergic, Nicotinic Alpha3Beta2
  • D(1A) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Dopamine D5 receptor
  • Dopamine receptor
  • Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1)
  • Histamine H1 receptor
  • Histamine H2 Receptor
  • Histamine H4 receptor
  • Imidazoline I1
  • Ionotropic glutamate receptor NMDA 1/2D
  • Kappa-type opioid receptor
  • Metabotropic glutamate receptor
  • Metabotropic glutamate receptor 2
  • Metabotropic glutamate receptor 4 (mGlu4)
  • Metabotropic glutamate receptor 6 (mGlu6)
  • Metabotropic glutamate receptor 8 (mGlu8)
  • Monoamine transporters; serotonin & dopamine
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Neuronal acetylcholine receptor
  • Neuronal acetylcholine receptor subunit alpha-4
  • Neuronal acetylcholine receptor; alpha2/beta2
  • Oxytocin receptor
  • Serotonin (5-HT) receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • Sodium-dependent noradrenaline transporter
  • Vasopressin V1b receptor
  • Vasopressin V2 receptor (V2)
570000000
  • L-homocysteine sulfinic acid