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Compound Name:

Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically

Compound Name (alphabetical)	Binding Targets	Enz. Inhib. Data							ITC Data	Alternate Compound Names
		Ki	IC50	Kd	EC50	Koff	Kon	Other
BDBM50171290	5-Hydroxytryptamine receptor 7 (5-HT7) 5-hydroxytryptamine receptor 1B 5-hydroxytryptamine receptor 1D 5-hydroxytryptamine receptor 2A 5-hydroxytryptamine receptor 2C 5-hydroxytryptamine receptor 3A 5-hydroxytryptamine receptor 4 (5-HT4) ADORA3 ATP-sensitive inward rectifier potassium channel 1 AVPR1A Adenosine receptor A1 Adenosine receptor A2 Alpha-1A adrenergic receptor Alpha-2A adrenergic receptor Alpha-2B adrenergic receptor Alpha-2C adrenergic receptor Angiotensin II AT2 Angiotensin II receptor Benzodiazepine central Benzodiazepine peripheral Beta-1 adrenergic receptor Beta-2 adrenergic receptor and beta-3 adrenergic receptor CHRM5 Calcitonin gene-related peptide (CGRP alpha) Calcium channel (DHP) Calcium channel (Type L) Cannabinoid receptor 1 Cannabinoid receptor 2 Chloride channel, TBOB Cholecystokinin receptor Cysteinyl leukotriene receptor 1 D(1A) dopamine receptor D(2) dopamine receptor D(3) dopamine receptor Disintegrin and metalloproteinase domain-containing protein 17 Dopamine D5 receptor Dopamine receptors; D2 & D4 EDNRB Endothelin-1 receptor GALANIN GRIA3 GRIK1 GRPR Gamma-aminobutyric acid type B receptor subunit 1 Glucocorticoid receptor Glutamate receptor ionotropic, NMDA 1 Glycine, non-strychnine HTR6 Histamine H1 receptor Histamine H2 Receptor Histamine receptor (H3) Imidazoline receptor 1 (I1R) Kappa-type opioid receptor Leukotriene 2 Melatonin receptor Muscarinic acetylcholine receptor M1 Muscarinic acetylcholine receptor M2 Muscarinic acetylcholine receptor M3 Muscarinic acetylcholine receptor M4 NMBR NT Neuromedin-K receptor Neuropeptide Y receptor type 1 Neuropeptide Y receptor type 2 Nociceptin/mu opioid receptor P2X purinoceptor 1 Platelet activating factor receptor Potassium Channel (Ca2+ dependent) Prostaglandin G/H synthase (cyclooxygenase) Purinergic receptor P2Y1 SOMATOSTATIN Serotonin (5-HT) receptor Sigma-1 Substance-K receptor Substance-P receptor VIP peptides Vasopressin V2 receptor (V2) Voltage-gated calcium channel subunit alpha Cav2.2 Voltage-gated potassium channel Voltage-gated sodium channel subunit alpha Nav1.1 (Nav1.1) Voltage-gated sodium channel subunit alpha Nav1.2 (Nav1.2)	88	0	0	0	0	0	0	0	5-(4-Bromo-phenyl)-1-(2,4-dichloro-phenyl)-4-ethyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide CHEMBL189676 SR 147778