BDBM104477 US8575186, 240/241::US8575186, 257
SMILES: COc1cc(cc2c3C4CCC(Cc3n(C)c12)N4)S(=O)(=O)n1ccc2ccccc12
InChI Key: InChIKey=MYAKLRIXBOSQBL-UHFFFAOYSA-N
Data: 2 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 6 (Homo sapiens (Human)) | BDBM104477 (US8575186, 240/241 | US8575186, 257) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Albany Molecular Research, Inc. US Patent | Assay Description The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ... | US Patent US8575186 (2013) BindingDB Entry DOI: 10.7270/Q2BR8QTS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 6 (Homo sapiens (Human)) | BDBM104477 (US8575186, 240/241 | US8575186, 257) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.850 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Albany Molecular Research, Inc. US Patent | Assay Description The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ... | US Patent US8575186 (2013) BindingDB Entry DOI: 10.7270/Q2BR8QTS | |||||||||||
More data for this Ligand-Target Pair |