null
SMILES: C[C@H]1CCCN1C1CCN(CC1)c1ccc(cc1)N1CCC2(CCN(CC2)S(=O)(=O)c2ccccc2)C1=O
InChI Key: InChIKey=JYGAXAVLOAJTOP-DEOSSOPVSA-N
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Macaca mulatta (Rhesus macaque)) | BDBM108309 (US8604046, 89) | UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Sanofi US Patent | Assay Description The compounds of this invention have been demonstrated to displace [3H]- methylhistamine radioligand binding to mammalian cell membranes expressing r... | US Patent US8604046 (2013) BindingDB Entry DOI: 10.7270/Q2W957TB | |||||||||||
More data for this Ligand-Target Pair |