BDBM136369 US8865750, CCG- 203780

SMILES: BrC1=CC(=O)N(Cc2ccccc2)C1=O

InChI Key: InChIKey=LLBVECSKMXUDOT-UHFFFAOYSA-N

Data: 2 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 136369   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Regulator of G-protein signaling 8 (Homo sapiens (Human))	BDBM136369 (US8865750, CCG- 203780) Show SMILES BrC1=CC(=O)N(Cc2ccccc2)C1=O |t:1| Show InChI InChI=1S/C11H8BrNO2/c12-9-6-10(14)13(11(9)15)7-8-4-2-1-3-5-8/h1-6H,7H2	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	US Patent	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
The Regents of The University of Michigan; The University of Bath US Patent					Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...				US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC
					More data for this Ligand-Target Pair
Regulator of G-protein signaling 4 (Homo sapiens (Human))	BDBM136369 (US8865750, CCG- 203780) Show SMILES BrC1=CC(=O)N(Cc2ccccc2)C1=O |t:1| Show InChI InChI=1S/C11H8BrNO2/c12-9-6-10(14)13(11(9)15)7-8-4-2-1-3-5-8/h1-6H,7H2	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase MCE PC cid PC sid UniChem	US Patent	n/a	n/a	3.20E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Regents of The University of Michigan; The University of Bath US Patent					Assay Description FCPIA Characterization of RGS Inhibitory Activity: CCG-50014 (FIG. 1) was originally identified as a potential inhibitor of RGS8 and RGS16 in a polyp...				US Patent US8865750 (2014) BindingDB Entry DOI: 10.7270/Q20000TC
					More data for this Ligand-Target Pair