BDBM186927 US9079895, 19s
SMILES: C(CN1CCO[C@H](COc2ccccc2)C1)N1CCc2ccccc12
InChI Key: InChIKey=ZKTUDHGKQCWRDH-FQEVSTJZSA-N
Data: 13 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 1A (5HT1A) (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dopamine D4 receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 132 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D(2) dopamine receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 342 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 7 (5HT7) (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 468 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1D (5HT1D) (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 590 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2A (5HT2A) (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | PDB UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 817 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dopamine D1 receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 1.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2B (5HT2B) (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 1.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1D adrenergic receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 2.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A adrenergic receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 2.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dopamine D3 receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 2.83E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 2C (5HT2C) (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 6.74E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1B adrenergic receptor (Mus musculus (Mouse)) | BDBM186927 (US9079895, 19s) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 7.21E+3 | n/a | n/a | n/a | n/a | n/a | n/a | 7.4 | n/a |
University of Dundee US Patent | Assay Description The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.un... | US Patent US9079895 (2015) BindingDB Entry DOI: 10.7270/Q2D7996K | |||||||||||
More data for this Ligand-Target Pair |