BDBM196929 US9212196, Derivative 25
SMILES: N[C@H](CCP(O)(=O)C(O)c1ccc(SCC(O)=O)c(c1)[N+]([O-])=O)C(O)=O
InChI Key: InChIKey=ZDPGMBDQVVWLAD-UOGPZTOASA-N
Data: 3 EC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 4 (mGlu4) (Rattus norvegicus (Rat)) | BDBM196929 (US9212196, Derivative 25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 7 (mGlu7) (Rattus norvegicus (Rat)) | BDBM196929 (US9212196, Derivative 25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.52E+4 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 8 (mGlu8) (Rattus norvegicus (Rat)) | BDBM196929 (US9212196, Derivative 25) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | n/a | n/a | 1.15E+4 | n/a | n/a | n/a | n/a |
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE US Patent | Assay Description Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ... | US Patent US9212196 (2015) BindingDB Entry DOI: 10.7270/Q28G8JJR | |||||||||||
More data for this Ligand-Target Pair |