BDBM200909 US9233946, 8
SMILES: CC(C)c1ccc2sc(c(C)c2c1)S(=O)(=O)Nc1nc(C)c(s1)C(O)=O
InChI Key: InChIKey=ZQESQZGRGLZODB-UHFFFAOYSA-N
Data: 1 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3) (Homo sapiens (Human)) | BDBM200909 (US9233946, 8) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 610 | n/a | n/a | n/a | n/a | n/a | n/a |
KANCERA AB US Patent | Assay Description Method A: The kinase activity of the bi-functional enzyme is readily quantified based on the production of F-2,6-P2 as described by Van Schaftingen e... | US Patent US9233946 (2016) BindingDB Entry DOI: 10.7270/Q2V123KB | |||||||||||
More data for this Ligand-Target Pair |