BDBM210829 US9290463, B
SMILES: Cn1c(=O)cnn(CCCCN2CCN(CC2)c2cccc(I)n2)c1=O
InChI Key: InChIKey=WSJDMNAJKWFILG-UHFFFAOYSA-N
Data: 1 KI
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-HT1A/ 5-HT2c (Homo sapiens (Human)) | BDBM210829 (US9290463, B) | PDB KEGG UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 5.5 | -10.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 4 |
The Trustees of Columbia University in the City of New York US Patent | Assay Description Preparation of Membrane Fractions from CHO-h5-HT1A Cells. Membranes from CHO cells stably expressing the human 5-HT1A receptor at a density of 8 pmol... | US Patent US9290463 (2016) BindingDB Entry DOI: 10.7270/Q2MS3RK0 | |||||||||||
More data for this Ligand-Target Pair |