BDBM21361 (5S)-5-Ethyl-3-methyl-5-phenyl-2,4-imidazolidinedione::(5S)-5-ethyl-3-methyl-5-phenylimidazolidine-2,4-dione::Mephenytoin, D-::S-Mephenytoin::S-mephentoin
SMILES: CC[C@]1(NC(=O)N(C)C1=O)c1ccccc1
InChI Key: InChIKey=GMHKMTDVRCWUDX-LBPRGKRZSA-N
Data: 5 IC50
Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Uridine-5'-diphosphoglucuronosyltransferase 1A1 (Homo sapiens (Human)) | BDBM21361 ((5S)-5-Ethyl-3-methyl-5-phenyl-2,4-imidazolidinedi...) | UniProtKB/SwissProt UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences | Assay Description Refer to Fisher et al., Drug Metab. Dispos., 28:560-566. | J Enzyme Inhib Med Chem 26: 386-93 (2011) Article DOI: 10.3109/14756366.2010.518965 BindingDB Entry DOI: 10.7270/Q2HQ3XS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uridine-5'-diphosphoglucuronosyltransferase 1A4 (Homo sapiens (Human)) | BDBM21361 ((5S)-5-Ethyl-3-methyl-5-phenyl-2,4-imidazolidinedi...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences | Assay Description Refer to Fisher et al., Drug Metab. Dispos., 28:560-566. | J Enzyme Inhib Med Chem 26: 386-93 (2011) Article DOI: 10.3109/14756366.2010.518965 BindingDB Entry DOI: 10.7270/Q2HQ3XS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uridine-5'-diphosphoglucuronosyltransferase 2B10 (Homo sapiens (Human)) | BDBM21361 ((5S)-5-Ethyl-3-methyl-5-phenyl-2,4-imidazolidinedi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences | Assay Description Refer to Fisher et al., Drug Metab. Dispos., 28:560-566. | J Enzyme Inhib Med Chem 26: 386-93 (2011) Article DOI: 10.3109/14756366.2010.518965 BindingDB Entry DOI: 10.7270/Q2HQ3XS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uridine-5'-diphosphoglucuronosyltransferase 2B7 (Homo sapiens (Human)) | BDBM21361 ((5S)-5-Ethyl-3-methyl-5-phenyl-2,4-imidazolidinedi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences | Assay Description Refer to Fisher et al., Drug Metab. Dispos., 28:560-566. | J Enzyme Inhib Med Chem 26: 386-93 (2011) Article DOI: 10.3109/14756366.2010.518965 BindingDB Entry DOI: 10.7270/Q2HQ3XS4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Uridine-5'-diphosphoglucuronosyltransferase 1A6 (Homo sapiens (Human)) | BDBM21361 ((5S)-5-Ethyl-3-methyl-5-phenyl-2,4-imidazolidinedi...) | UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences | Assay Description Refer to Fisher et al., Drug Metab. Dispos., 28:560-566. | J Enzyme Inhib Med Chem 26: 386-93 (2011) Article DOI: 10.3109/14756366.2010.518965 BindingDB Entry DOI: 10.7270/Q2HQ3XS4 | |||||||||||
More data for this Ligand-Target Pair |